SCHEMBL20204555

SCHEMBL20204555

COC(=N)/C(C=O)=C\NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 1/20 0.47
ADH1C P00326 1/20 0.47
ADH1A P07327 1/20 0.47
ADH7 P40394 1/20 0.47
NR4A1 P22736 1/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
ATM Q13315 1/20 0.37
CA12 O43570 1/20 0.37
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20204557 0.77 ADH1B (0.33) ADH1BADH1CADH1AADH7MAPT
SCHEMBL28153270 0.74 ADH1B (0.57) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL20204574 0.73 MAPT (0.52) MAPTALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL20204556 0.71 ADH1B (0.36) ADH1BADH1CADH1AADH7MAPT
SCHEMBL10151057 0.71 ADH1B (0.53) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL21095759 0.71 ADH1B (0.44) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL28580835 0.71 ADH1B (0.53) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL23188929 0.70 ADH1B (0.57) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL22680702 0.70 CA1 (0.40) ADH1BADH1CADH1AADH7NR4A1
SCHEMBL627479 0.69 ADH1B (0.54) ADH1BADH1CADH1AADH7NR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096510-A1 HETEROARYLPHENOXY BENZAMIDE KAPPA OPIOID LIGANDS PFIZER INC. (US) 2018-05-31 WO disclosed