SCHEMBL20204557

SCHEMBL20204557

C=CC/N=C/C(=C/NCc1ccccc1)C(=N)OC

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 1/20 0.33
ADH1C P00326 1/20 0.33
ADH1A P07327 1/20 0.33
ADH7 P40394 1/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HSD17B10 Q99714 1/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
RAB9A P51151 2/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20204555 0.77 ADH1B (0.47) ADH1BADH1CADH1AADH7CA1
SCHEMBL20204556 0.70 ADH1B (0.36) ADH1BADH1CADH1AADH7CA1
SCHEMBL6467025 0.65 ADH1B (0.48) ADH1BADH1CADH1AADH7GAA
SCHEMBL21095759 0.65 ADH1B (0.44) ADH1BADH1CADH1AADH7CYP2D6
SCHEMBL18835308 0.65 ADH1B (0.44) ADH1BADH1CADH1AADH7GAA
SCHEMBL20204574 0.64 MAPT (0.52) GAACYP2D6MEN1KMT2AALDH1A1
SCHEMBL22680702 0.63 CA1 (0.40) ADH1BADH1CADH1AADH7CYP2C9
SCHEMBL627479 0.63 ADH1B (0.54) ADH1BADH1CADH1AADH7GAA
SCHEMBL21095906 0.62 ADH1B (0.44) ADH1BADH1CADH1AADH7GAA
SCHEMBL21095911 0.61 ALDH1A1 (0.54) ADH1BADH1CADH1AADH7CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096510-A1 HETEROARYLPHENOXY BENZAMIDE KAPPA OPIOID LIGANDS PFIZER INC. (US) 2018-05-31 WO disclosed