SCHEMBL20207796

SCHEMBL20207796

CC(C)Cc1ccc(CN)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.38
DAO P14920 1/20 0.35
LOXL2 Q9Y4K0 3/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
GPR84 Q9NQS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13327029 0.88 DAO (0.41) PARP1DAOKDM4EMAPTGABRA1
SCHEMBL2967282 0.80
SCHEMBL14012134 0.77 GABRA1 (0.35) PARP1DAOKDM4EGABRA1GABRB2
SCHEMBL20376636 0.77 DAO (0.35) PARP1DAOGABRA1GABRB2GPR84
SCHEMBL21324887 0.74 DAO (0.33) PARP1DAOKDM4EMAPTGPR84
SCHEMBL14754136 0.73
SCHEMBL20801759 0.73 LOXL2 (0.33) LOXL2
SCHEMBL9878781 0.69
SCHEMBL24881442 0.67 PABPC1 (0.47) PARP1DAOKDM4EGABRA1GABRB2
SCHEMBL14012135 0.67 GABRA1 (0.35) PARP1DAOGABRA1GABRB2GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098208-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed