SCHEMBL20214599

SCHEMBL20214599

NC(=O)c1ccccc1[S+]([O-])C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 3/20 0.42
MAPT P10636 3/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
METAP2 P50579 1/20 0.40
CTNNB1 P35222 1/20 0.40
BCAT2 O15382 1/20 0.39
PDK2 Q15119 1/20 0.39
LMNA P02545 2/20 0.37
GAA P10253 2/20 0.36
USP2 O75604 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
PARP1 P09874 1/20 0.36
NPC1 O15118 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
RAB9A P51151 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055459 0.82 KDM4E (0.42) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL6228527 0.76 KDM4E (0.47) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL1743540 0.73 BCAT2 (0.44) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL8042279 0.72 MAPT (0.42) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL8055106 0.71 ALDH1A1 (0.42) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL8054028 0.71 IRAK4 (0.46) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL11524577 0.71 ALDH1A1 (0.38) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL1001688 0.71 ALOX15 (0.38) ALDH1A1MAPTTSHRPDK2GAA
SCHEMBL8057920 0.70 CYP3A4 (0.47) KDM4EALDH1A1HPGDMAPTTSHR
SCHEMBL25087672 0.69 TSHR (0.39) ALDH1A1TSHRPDK2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056999-A9 ENANTIOMERICALLY ENRICHED ARYLOAZOL- 2 -YL CYANOETHYLAMINO PARACITICIDAL COMPOUNDS MERIAL LIMITED (US) 2018-06-07 WO disclosed