SCHEMBL20217846

SCHEMBL20217846

CC(O)CC1COCC(C)N1c1ccc(C(=N)c2cc(C(=O)NC(c3ccccn3)C3CCCC3)ccc2N)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.49
TTK P33981 7/20 0.49
AURKB Q96GD4 7/20 0.49
INCENP Q9NQS7 7/20 0.49
KCNK3 O14649 1/20 0.33
SLC6A9 P48067 1/20 0.32
WDR5 P61964 5/20 0.31
HTR3A P46098 2/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
BRD4 O60885 2/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217484 0.86 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217662 0.84 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPKCNK3
SCHEMBL20217579 0.83 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217446 0.80 CYP3A4 (0.53) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217956 0.80 CYP3A4 (0.48) CYP3A4TTKAURKBINCENPKCNK3
SCHEMBL20217481 0.79 ALDH1A1 (0.38) MEN1ALDH1A1KMT2A
SCHEMBL20217912 0.78 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217549 0.77 CYP3A4 (0.49) CYP3A4TTKAURKBINCENPHTR3A
SCHEMBL20217462 0.77 MAPT (0.38) CYP3A4ALDH1A1MAPK1KMT2A
SCHEMBL20217145 0.77 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed