SCHEMBL20239303

SCHEMBL20239303

CSc1nc(CNC(=O)OC(C)(C)C)cc(Oc2ccc(CS(N)(=O)=O)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 1/20 0.41
LMNA P02545 2/20 0.39
TSHR P16473 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA1 P00915 9/20 0.39
CA2 P00918 9/20 0.39
CA12 O43570 7/20 0.39
CA9 Q16790 7/20 0.39
MAPT P10636 2/20 0.38
DYRK1A Q13627 1/20 0.35
GRM2 Q14416 1/20 0.34
KDM4A O75164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20259075 0.88 DGAT2 (0.43) DGAT2CA1CA2CA12CA9
SCHEMBL20239318 0.88 LMNA (0.45) DGAT2LMNATSHRNPSR1CA1
SCHEMBL18249768 0.86 DGAT2 (0.44) DGAT2LMNACA1CA2CA12
SCHEMBL20259162 0.86 DGAT2 (0.42) DGAT2CA1CA2CA12CA9
SCHEMBL20259248 0.85 DGAT2 (0.41) DGAT2CA1CA2CA12CA9
SCHEMBL20239235 0.73 DGAT2 (0.44) DGAT2LMNANPSR1MEN1KMT2A
SCHEMBL20239312 0.73 DGAT2 (0.47) DGAT2LMNACA1CA2CA9
SCHEMBL20239264 0.73 DGAT2 (0.45) DGAT2LMNATSHRNPSR1MAPT
SCHEMBL20239187 0.73 LMNA (0.41) DGAT2LMNATSHRNPSR1CA1
SCHEMBL20239327 0.72 DGAT2 (0.44) DGAT2LMNATSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107635975-B DGAT2 inhibitors 伊莱利利公司 2020-07-24 CN disclosed
EP-3298001-B1 DGAT2 INHIBITORS LILLY CO ELI (US) 2020-05-13 EP disclosed
US-10053429-B2 DGAT2 inhibitors ELI LILLY AND COMPANY (US) 2018-08-21 US disclosed
US-20180162825-A1 NOVEL DGAT2 INHIBITORS ELI LILY AND COMPANY (US) 2018-06-14 US disclosed
US-20180162825-A1 NOVEL DGAT2 INHIBITORS ELI LILY AND COMPANY (US) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180162825-A1 NOVEL DGAT2 INHIBITORS DGAT2, DGAT1, LCAT DGAT2 1/4885LMNA 2022/4885TSHR 777/4885
US-10053429-B2 DGAT2 inhibitors DGAT2, DGAT1, LCAT DGAT2 1/4885LMNA 1722/4885TSHR 690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.