SCHEMBL20249755

SCHEMBL20249755

Nc1ccc(-n2ccc(N)n2)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
GABRP O00591 2/20 0.34
GABRD O14764 2/20 0.34
GABRA1 P14867 2/20 0.34
GABRB1 P18505 2/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA5 P31644 2/20 0.34
GABRA3 P34903 2/20 0.34
GABRA2 P47869 2/20 0.34
GABRB2 P47870 2/20 0.34
GABRA4 P48169 2/20 0.34
GABRE P78334 2/20 0.34
GABRA6 Q16445 2/20 0.34
GABRG1 Q8N1C3 2/20 0.34
GABRG3 Q99928 2/20 0.34
GABRQ Q9UN88 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13662722 0.83 ELANE (0.38) NOS3NOS2CHRNB2CHRNA4SMN1; SMN2
SCHEMBL20242125 0.83 POLB (0.50) CHRNB2CHRNA4PIK3CDMAPT
SCHEMBL20390956 0.83
SCHEMBL31052478 0.79 DHFR (0.44) PIK3CDMAPTMAP4K4KCNH2MINK1
SCHEMBL20390801 0.79 CHRNB2 (0.41) CHRNB2CHRNA4PIK3CDNNMTKCNH2
SCHEMBL31316711 0.79 CHRNB2 (0.41) CHRNB2CHRNA4PIK3CDNNMTKCNH2
SCHEMBL13623576 0.79 PDE10A (0.30)
SCHEMBL20242304 0.79 NNMT (0.39) NNMTMAPTKCNH2MKNK1
SCHEMBL13615877 0.79 CHRNA7 (0.33)
SCHEMBL20250065 0.79 KCNH2 (0.38) MAPTHDAC6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018107056-A1 1,3-SUBSTITUED PYRAZOLE COMPOUNDS USEFUL FOR REDUCTION OF VERY LONG CHAIN FATTY ACIC LEVELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2018-06-14 WO disclosed