SCHEMBL20255437

SCHEMBL20255437

O=C(O)C1CCN(Cc2ccc(I)nc2)C1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 11/20 0.54
S1PR1 P21453 2/20 0.54
S1PR4 O95977 1/20 0.54
S1PR3 Q99500 1/20 0.54
CD274 Q9NZQ7 5/20 0.51
PDCD1 Q15116 4/20 0.51
LTA4H P09960 3/20 0.47
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037857 0.92 L3MBTL1 (0.51) S1PR5S1PR1S1PR4S1PR3LTA4H
SCHEMBL20037434 0.84 S1PR5 (0.54) S1PR5S1PR1S1PR4S1PR3CD274
SCHEMBL18291640 0.84 S1PR5 (0.57) S1PR5S1PR1S1PR4S1PR3CD274
SCHEMBL20037684 0.83 NPC1 (0.55) LTA4HKMT2A
SCHEMBL20249155 0.81 S1PR5 (0.54) S1PR5S1PR1S1PR4S1PR3CD274
SCHEMBL20255702 0.81 ALDH1A1 (0.47) CD274PDCD1LTA4HKMT2A
SCHEMBL20255353 0.81 ALDH1A1 (0.47) CD274PDCD1LTA4HKMT2A
SCHEMBL20037837 0.80 LTA4H (0.49) LTA4HKMT2A
SCHEMBL16193062 0.79 HRH3 (0.48) LTA4HKMT2A
SCHEMBL20037952 0.79 HRH3 (0.48) LTA4HKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 S1PR5 2141/4885S1PR1 2509/4885S1PR4 2204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.