SCHEMBL20257512

SCHEMBL20257512

COC(=O)N[C@@H](CCc1cccnc1)C(=O)NCCCCN1C(=N)NC(c2ccccc2)(c2ccccc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.38
EPHX2 P34913 1/20 0.38
PTAFR P25105 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 1/20 0.37
CTSL P07711 4/20 0.37
CTSB P07858 4/20 0.37
FES P07332 1/20 0.36
RET P07949 1/20 0.36
MARK3 P27448 1/20 0.36
TYK2 P29597 1/20 0.36
FLT4 P35916 1/20 0.36
SYK P43405 1/20 0.36
CLK2 P49760 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21553895 0.93 AKT1 (0.40) EPHX1EPHX2PTAFRL3MBTL1NPC1
SCHEMBL20257403 0.93 L3MBTL1 (0.43) L3MBTL1NPC1CHRNB2CHRNB4CHRNA3
SCHEMBL20257434 0.92 L3MBTL1 (0.40) L3MBTL1NPC1CHRNB2CHRNB4CHRNA3
SCHEMBL20257432 0.88 NPY1R (0.38) L3MBTL1NPC1CYP3A4FAAH
SCHEMBL20257514 0.87 CHRNB2 (0.42) L3MBTL1CTSLCHRNB2CHRNB4CHRNA3
SCHEMBL20241812 0.86 AKT1 (0.47) L3MBTL1NPC1CTSLCTSBCHRNB2
SCHEMBL21553986 0.86 AKT1 (0.42) L3MBTL1NPC1MMP9CYP3A4FAAH
SCHEMBL20257513 0.86 PTAFR (0.40) EPHX1EPHX2PTAFRFESRET
SCHEMBL20241617 0.86 AKT1 (0.46) L3MBTL1NPC1CTSLCTSBCHRNB2
SCHEMBL21553989 0.85 AKT1 (0.41) L3MBTL1NPC1MMP9CYP3A4FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018106519-A1 HETEROCYCLIC COMPOUNDS AS HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-06-14 WO disclosed