SCHEMBL20260359

SCHEMBL20260359

Cc1cc(N2CC(N3CCOCC3)C2)ccc1Nc1ncn(-c2cc(F)cc(F)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TTK P33981 11/20 0.44
P2RX7 Q99572 4/20 0.41
PIK3CA P42336 1/20 0.41
MAPK8 P45983 2/20 0.38
MAPK10 P53779 2/20 0.38
MAPK9 P45984 1/20 0.38
ACVR1 Q04771 1/20 0.36
TBK1 Q9UHD2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20260395 0.94 P2RX7 (0.39) TTKP2RX7PIK3CAMAPK8MAPK10
SCHEMBL18278673 0.89 MAPK8 (0.36) TTKP2RX7PIK3CAMAPK8MAPK10
SCHEMBL18277739 0.89 MAPK10 (0.36) TTKP2RX7PIK3CAMAPK8MAPK10
SCHEMBL20260363 0.84 TTK (0.44) TTKP2RX7PIK3CAACVR1
SCHEMBL20260939 0.84 P2RX7 (0.39) TTKP2RX7MAPK8MAPK10MAPK9
SCHEMBL20260924 0.84 MAPK8 (0.35) TTKMAPK8MAPK10MAPK9ACVR1
SCHEMBL20260873 0.83 MAPT (0.42) MAPK8MAPK10MAPK9
SCHEMBL20242649 0.83 MAPK14 (0.38) TTKMAPK8MAPK10MAPK9ACVR1
SCHEMBL18278851 0.83 MAPK8 (0.34) TTKMAPK8MAPK10MAPK9ACVR1
SCHEMBL18278868 0.83 MAPK8 (0.34) TTKMAPK8MAPK10MAPK9ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018106646-A1 AMINOTRIAZOLES FOR THE TREATMENT OF DEMYELINATING DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2018-06-14 WO disclosed