SCHEMBL20274207

SCHEMBL20274207

O=C(CO)N1CCN(Cc2nc3cc(F)ccc3s2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.49
KCNH2 Q12809 3/20 0.47
GPR119 Q8TDV5 3/20 0.47
AKR1B1 P15121 3/20 0.45
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
AKR1A1 P14550 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NAAA Q02083 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DYRK1A Q13627 1/20 0.41
EPHX2 P34913 1/20 0.41
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20274201 0.86 EPHX2 (0.52) HDAC6AKR1B1NPC1RAB9AEPHX2
SCHEMBL20651340 0.86 HDAC6 (0.49) HDAC6KCNH2AKR1B1TP53L3MBTL1
SCHEMBL20274125 0.85 AKR1B1 (0.53) HDAC6AKR1B1AKR1A1L3MBTL1DYRK1A
SCHEMBL20274208 0.80 KCNH2 (0.43) HDAC6KCNH2GPR119AKR1B1AKR1A1
SCHEMBL20274151 0.79 FAAH (0.48) AKR1B1MAPTTP53NPC1RAB9A
SCHEMBL15708163 0.78 HDAC6 (0.46) HDAC6KCNH2GPR119AKR1B1AKR1A1
SCHEMBL20274161 0.74 KCNH2 (0.52) KCNH2TP53NPC1RAB9ACYP2D6
SCHEMBL20274164 0.74 KCNH2 (0.42) KCNH2GPR119AKR1B1AKR1A1DYRK1A
SCHEMBL23336086 0.73 FAAH (0.57) CYP2D6CYP2C9ALOX15TSHRCYP2C19
SCHEMBL20964520 0.71 AKR1B1 (0.52) HDAC6AKR1B1AKR1A1L3MBTL1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428162-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC (US) 2021-05-05 EP disclosed
EP-2922845-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC (US) 2018-06-20 EP disclosed