SCHEMBL20274814

SCHEMBL20274814

CC(C)(C)OC(=O)N[C@H](CO)Cc1ccc(-c2cnc(NCc3ccc4ccccc4c3)cn2)cc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 12/20 0.61
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
CTSB P07858 1/20 0.43
ATM Q13315 1/20 0.43
PTPN1 P18031 2/20 0.38
SCN9A Q15858 1/20 0.38
CYP3A4 P08684 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL308330 0.88 TPH1 (0.66) TPH1CTSSCTSKCTSBPTPN1
SCHEMBL308331 0.88 TPH1 (0.66) TPH1CTSSCTSKCTSBPTPN1
SCHEMBL31584190 0.80 CTSS (0.61) CTSSCTSKCTSBATMPTPN1
SCHEMBL7353984 0.80 CTSS (0.61) CTSSCTSKCTSBATMPTPN1
SCHEMBL9266214 0.78 CTSB (0.52) CTSSCTSKCTSBATMPTPN1
SCHEMBL15315375 0.78 TPH1 (0.68) TPH1
SCHEMBL308167 0.76 TPH1 (1.00) TPH1
SCHEMBL1531589 0.74 CTSS (0.62) CTSSCTSKCTSBATMPTPN1
SCHEMBL1531592 0.74 CTSS (0.62) CTSSCTSKCTSBATMPTPN1
SCHEMBL15521493 0.74 CTSS (0.62) CTSSCTSKCTSBATMPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2386547-B1 Multicyclic amino acid derivatives and methods of their use LEXICON PHARMACEUTICALS INC (US) 2018-06-20 EP disclosed