SCHEMBL20301032

SCHEMBL20301032

CC1(C)N=C(c2ccc3ccccc3n2)c2ccc(Cl)cc2C1(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.38
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
PDK2 Q15119 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 2/20 0.34
CNR1 P21554 1/20 0.34
ACP1 P24666 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
NR4A2 P43354 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX12 P18054 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20300747 0.91 AR (0.38) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20301881 0.88 AR (0.38) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20300854 0.87 AR (0.38) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20301183 0.86 PDK2 (0.34) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20301260 0.85 NPC1 (0.39) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20300741 0.85 PDK2 (0.33) KDM4EPDK2TDP1ACP1ALDH1A1
SCHEMBL4514362 0.79 TDP2 (0.38) CYP1A2CNR1HPGDCYP2D6
SCHEMBL20301261 0.79 AR (0.43) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20301474 0.75 NPC1 (0.40) ARKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20300813 0.75 HSD11B1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO claimed
WO-2018116072-A1 HETEROCYCLIC COMPOUNDS PI INDUSTRIES LTD. (IN) 2018-06-28 WO disclosed