SCHEMBL20307752

SCHEMBL20307752

COC(=O)c1nn(C)c(-c2ccc(CO[Si](C)(C)C(C)(C)C)cc2)c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.33
GRM5 P41594 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
AURKA O14965 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
HTT P42858 1/20 0.31
FAAH O00519 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16258908 0.83 SMN1; SMN2 (0.36) SMN1; SMN2MAPTMEN1LMNAKMT2A
SCHEMBL10140470 0.78 KCNA3 (0.32) SMN1; SMN2MAPTMEN1KMT2AALDH1A1
SCHEMBL1313112 0.73 LOXL2 (0.51) SMN1; SMN2MAPTKDM4EMEN1LMNA
SCHEMBL505474 0.69 TACR1 (0.38) MAPTLMNAKMT2AALDH1A1HTT
SCHEMBL9435638 0.68 CYP4F2 (0.50) SMN1; SMN2MAPTKDM4ELMNAKMT2A
SCHEMBL20742521 0.68 XDH (0.42) SMN1; SMN2LMNAFAAH
SCHEMBL6472720 0.67 KDM4E (0.43) MAPTKDM4EMEN1KMT2AALDH1A1
SCHEMBL10172623 0.67 ALDH1A1 (0.52) SMN1; SMN2MAPTKMT2AALDH1A1HPGD
SCHEMBL11298531 0.67 SMN1; SMN2 (0.61) SMN1; SMN2MAPTMEN1LMNAKMT2A
SCHEMBL8128802 0.67 KDM4E (0.44) SMN1; SMN2MAPTKDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805939-B1 Heterocyclic compounds as factor IXA inhibitors. MERCK SHARP & DOHME (US) 2018-06-27 EP disclosed