SCHEMBL2032499

SCHEMBL2032499

NCC(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.56
ITGB3 P05106 2/20 0.54
ITGA2B P08514 2/20 0.54
MME P08473 1/20 0.52
ACE P12821 5/20 0.52
AOC3 Q16853 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CTSC P53634 2/20 0.50
ECE1 P42892 1/20 0.50
LMNA P02545 1/20 0.50
NAALAD2 Q9Y3Q0 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16983210 1.00 MMP2 (0.56) MMP2ITGB3ITGA2BMMEACE
SCHEMBL2032501 1.00 MMP2 (0.56) MMP2ITGB3ITGA2BMMEACE
SCHEMBL29630808 0.99 MMP2 (0.55) MMP2ITGB3ITGA2BMMEACE
SCHEMBL30051999 0.95 CTSB (0.55) MMP2ITGB3ITGA2BMMEACE
SCHEMBL30051480 0.95 CTSB (0.55) MMP2ITGB3ITGA2BMMEACE
SCHEMBL23142823 0.95 CTSB (0.55) MMP2ITGB3ITGA2BMMEACE
SCHEMBL23142822 0.95 CTSB (0.55) MMP2ITGB3ITGA2BMMEACE
SCHEMBL30997458 0.91 QRFPR (0.54) MMP2ITGB3ITGA2BMME
SCHEMBL30439820 0.91 OPRD1 (0.52) ITGB3ITGA2BMMECTSCLMNA
SCHEMBL30439797 0.91 OPRD1 (0.52) ITGB3ITGA2BMMECTSCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2995 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137795-A1 EXATECAN IMMUNOCONJUGATES IMMUNOME INC (US) 2026-05-21 US claimed
US-12622975-B2 Peptide-conjugated prodrugs BRANDEIS UNIVERSITY (US) 2026-05-12 US claimed
US-20260077056-A1 LINKER-PAYLOAD COMPOUND, CONJUGATES AND APPLICATIONS THEREOF GENEQUANTUM HEALTHCARE SUZHOU CO LTD (CN) 2026-03-19 US claimed
EP-4695258-A1 BENZOPORPHYRIN ANALOGS, CONJUGATES, AND METHODS OF USE THEREOF Nira Biosciences, Inc. (US) 2026-02-18 EP claimed
EP-4684807-A1 LINKER AND USE THEREOF IN LIGAND DRUG CONJUGATE Duality Biologics (Shanghai) Co., Ltd. (CN) 2026-01-28 EP claimed
EP-4684805-A1 SELECTIVE ANTIBODY-DRUG CONJUGATES FOR TARGETED CANCER THERAPY Universitätsmedizin der Johannes Gutenberg-Universität Mainz (DE) 2026-01-28 EP claimed
US-20260021193-A1 IMMUNOCONJUGATES AND METHODS IMMUNOME INC (US) 2026-01-22 US claimed
EP-4655006-A2 EXATECAN IMMUNOCONJUGATES Immunome, Inc. (US) 2025-12-03 EP claimed
EP-4648799-A1 LIGAND-DRUG CONJUGATES Sun Pharma Advanced Research Company Ltd (IN) 2025-11-19 EP claimed
US-20250332272-A1 PREPARATION METHOD FOR DRUG LINKER CONJUGATE AND INTERMEDIATE THEREOF MEDILINK THERAPEUTICS SUZHOU CO LTD (CN) 2025-10-30 US claimed
WO-2022150642-A1 ANTI-INTERLEUKIN 36 RECEPTOR (IL-36R) THERAPY FOR HIDRADENITIS SUPPURATIVA ANAPTYSBIO, INC. (US) 2022-07-14 WO claimed
WO-2022150644-A1 ANTI-INTERLEUKIN 36 RECEPTOR (IL-36R) THERAPY FOR ACNE ANAPTYSBIO, INC. (US) 2022-07-14 WO claimed
US-20220211863-A1 COMPOUNDS AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2022-07-07 US claimed
US-20220193069-A1 CAMPTOTHECIN PEPTIDE CONJUGATES SEAGEN INC (US) 2022-06-23 US claimed
WO-2022112356-A1 TREATMENT OF CANCER INNATE PHARMA (FR) 2022-06-02 WO claimed
WO-2022078524-A2 SPECIFIC CONJUGATION OF AN ANTIBODY HANGZHOU DAC BIOTECH CO., LTD. (CN) 2022-04-21 WO claimed
WO-2022026832-A9 ANTI-INTERLEUKIN 36 RECEPTOR (IL-36R) THERAPY FOR ICHTHYOSIS ANAPTYSBIO, INC. (US) 2022-03-24 WO claimed
WO-2022026832-A1 ANTI-INTERLEUKIN 36 RECEPTOR (IL-36R) THERAPY FOR ICHTHYOSIS ANAPTYSBIO, INC. (US) 2022-02-03 WO claimed
WO-2022026829-A1 ANTI-INTERLEUKIN 36 RECEPTOR (IL-36R) THERAPY FOR SKIN TOXICITY ANAPTYSBIO, INC. (US) 2022-02-03 WO claimed
US-20150291659-A1 SOLOMONAMIDE ANALOGUE COMPOUNDS, PHARMACEUTICALS CONTAINING SOLOMONAMIDE ANALOGUE COMPOUNDS, AND PROCESSES FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2015-10-15 US claimed