SCHEMBL20329554

SCHEMBL20329554

Cc1cccc(C(F)(F)F)c1N(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
CYP1A2 P05177 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HSD11B1 P28845 2/20 0.35
AXL P30530 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
P2RX7 Q99572 1/20 0.34
AR P10275 4/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.33
ACP1 P24666 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25722706 0.87 TDP1 (0.40) CYP1A2TDP1CYP3A4ALOX15TSHR
SCHEMBL25491239 0.81 GABRA1 (0.52) GABRA1GABRB2CYP1A2TDP1TSHR
SCHEMBL25005922 0.79 HSD11B1 (0.38) CYP1A2TDP1CYP3A4ALOX15TSHR
SCHEMBL24497694 0.78 PTK2 (0.46) CYP1A2TDP1CYP3A4TSHRAXL
SCHEMBL22662731 0.78 CYP1A2 (0.35) CYP1A2TDP1CYP3A4ALOX15TSHR
SCHEMBL22662730 0.78 TSHR (0.35) CYP1A2TDP1CYP3A4ALOX15TSHR
SCHEMBL1107763 0.77 CYP2A6 (0.45) CYP1A2TDP1ALOX15TSHRHSD17B10
SCHEMBL24655960 0.75 AR (0.41) CYP3A4ALOX15TSHRMAPK1HSD17B10
SCHEMBL19130451 0.75 P2RX7 (0.46) GABRA1GABRB2CYP1A2TDP1CYP3A4
Hydrochloric Acid SCHEMBL2857487 0.74 CYP2A6 (0.43) CYP1A2TDP1CYP3A4ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018118947-A1 THIENOPYRROLE DERIVATIVES FOR USE IN TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. (US) 2018-06-28 WO disclosed