SCHEMBL20333380

SCHEMBL20333380

CCOC(Cc1ccc(NC(=O)c2cccs2)cc1)(C(=O)O)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.60
MEN1 O00255 8/20 0.60
TP53 P04637 3/20 0.60
ALDH1A1 P00352 1/20 0.60
NPC1 O15118 8/20 0.59
RAB9A P51151 8/20 0.59
SMN1; SMN2 Q16637 5/20 0.59
TDP1 Q9NUW8 2/20 0.57
MAPT P10636 4/20 0.54
LMNA P02545 2/20 0.54
GFER P55789 1/20 0.54
KDM4E B2RXH2 2/20 0.54
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
HTT P42858 1/20 0.51
CASP3 P42574 1/20 0.51
CASP2 P42575 1/20 0.51
POLB P06746 2/20 0.51
RECQL P46063 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22216671 0.86 MEN1 (0.60) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL22216493 0.86 MEN1 (0.60) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL20347168 0.83 MEN1 (0.56) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL20333771 0.83 NPC1 (0.56) KMT2AMEN1NPC1RAB9ASMN1; SMN2
SCHEMBL308069 0.79 NPC1 (0.75) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL20334149 0.75 RAB9A (0.49) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL29684837 0.75 RAB9A (0.71) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL1685916 0.74 SMN1; SMN2 (0.48) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL1929165 0.73 NPC1 (0.85) KMT2AMEN1TP53ALDH1A1NPC1
SCHEMBL8868420 0.72 NPC1 (0.73) KMT2AMEN1TP53ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018119284-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF CALITHERA BIOSCIENCES, INC. (US) 2018-06-28 WO disclosed