SCHEMBL308069

SCHEMBL308069

CCc1ccc(NC(=O)c2cccs2)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.75
RAB9A P51151 8/20 0.75
MEN1 O00255 8/20 0.75
KMT2A Q03164 8/20 0.75
TDP1 Q9NUW8 2/20 0.75
TP53 P04637 4/20 0.71
ALDH1A1 P00352 2/20 0.71
SMN1; SMN2 Q16637 7/20 0.70
MAPT P10636 6/20 0.66
NFKB1 P19838 1/20 0.66
NFKB2 Q00653 1/20 0.66
RELA Q04206 1/20 0.66
LMNA P02545 2/20 0.65
HTT P42858 2/20 0.65
GFER P55789 1/20 0.65
CASP3 P42574 1/20 0.64
CASP2 P42575 1/20 0.64
KDM4E B2RXH2 2/20 0.63
POLB P06746 3/20 0.63
USP2 O75604 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12443652 0.84 MAPK1 (0.67) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL8868420 0.83 NPC1 (0.73) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL8868426 0.83 NPC1 (0.73) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL29684837 0.82 RAB9A (0.71) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL12495837 0.82 NPC1 (1.00) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL22804218 0.82 NPC1 (0.83) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL8771200 0.82 NPC1 (0.89) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL19392293 0.82 NPC1 (0.89) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL16298403 0.81 NPC1 (0.80) NPC1RAB9AMEN1KMT2ATDP1
SCHEMBL2063276 0.80 NPC1 (0.86) NPC1RAB9AMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4738766-A2 DATA TRANSMISSION CONTROL METHOD AND SYSTEM, AND FIRST END, DEVICE AND READABLE STORAGE MEDIUM Huang, Jianfang (CN) 2026-05-06 EP disclosed
US-20250069572-A1 SCALE SHIFTING AND VOLUME ADJUSTMENT METHODS, APPARATUS, AND DEVICE RINGWAY TECH (JIANGSU) CO., LTD. (CN) 2025-02-27 US disclosed
US-20240029765-A1 Methods for Programming and Accessing Resistive Change Elements Using Neutral Voltage Conditions NANTERO, INC. (US) 2024-01-25 US disclosed
US-11817171-B2 Devices for providing neutral voltage conditions for resistive change elements in resistive change element arrays NANTERO, INC. (US) 2023-11-14 US disclosed
CN-110291148-B Rubber composition for conveyor belt, method for producing rubber composition for conveyor belt, and belt conveyor 横滨橡胶株式会社 2022-06-21 CN disclosed
US-20220028435-A1 Devices for Providing Neutral Voltage Conditions for Resistive Change Elements in Resistive Change Element Arrays NANTERO, INC. (US) 2022-01-27 US disclosed
US-8410121-B2 Methods of treating pulmonary hypertension LEXICON PHARMACEUTICALS, INC. (US) 2013-04-02 US disclosed
US-8093291-B2 Methods of using and compositions comprising tryptophan hydroxylase inhibitors LEXICON PHARMACEUTICALS, INC. (US) 2012-01-10 US disclosed
US-8063057-B2 Multicyclic amino acid derivatives and methods of their use LEXICON PHARMACEUTICALS, INC. (US) 2011-11-22 US disclosed
EP-2386547-A1 Multicyclic amino acid derivatives and methods of their use Lexicon Pharmaceuticals, Inc. (US) 2011-11-16 EP disclosed
US-20110263601-A1 METHODS OF TREATING ULCERATIVE COLITIS LEXICON PHARMACEUTICALS, INC. 2011-10-27 US disclosed
US-8039086-B2 Bonding material, process for producing the same, and honeycomb structure made with the same NGK INSULATORS, LTD. (JP) 2011-10-18 US disclosed
WO-2011100285-A1 TRYPTOPHAN HYDROXYLASE INHIBITORS FOR THE TREATMENT OF METASTATIC BONE DISEASE LEXICON PHARMACEUTICALS, INC. (US) 2011-08-18 WO disclosed
WO-2011056916-A1 TRYPTOPHAN HYDROXYLASE INHIBITORS FOR THE TREATMENT OF CANCER LEXICON PHARMACEUTICALS, INC. (US) 2011-05-12 WO disclosed
US-20110112094-A1 Methods of Treating Pulmonary Hypertension TERSERA THERAPEUTICS LLC 2011-05-12 US disclosed
US-7875622-B2 administering to a patient A therapeutically effective amounts of an endothelin receptor antagonist e.g. ambrisentan, bosentan etc. and (S)-2-amino-3-(4-(2-amino-6-((R)-2,2,2-trifluoro-1-(3'-methoxybiphenyl-4-yl)ethoxy)pyrimidin-4-yl)phenyl)propanoic acid to treat pulmonary hypertension LEXICON PHARMACEUTICALS, INC. (US) 2011-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112094-A1 Methods of Treating Pulmonary Hypertension TPH1, TPH2, PTGIS NPC1 4278/4885RAB9A 3956/4885MEN1 2873/4885
US-20110263601-A1 METHODS OF TREATING ULCERATIVE COLITIS TPH2, TPH1, HNMT NPC1 4113/4885RAB9A 4199/4885MEN1 4840/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.