SCHEMBL20334149

SCHEMBL20334149

CCOC(=O)C(Cc1ccc(NC(=O)c2cccs2)cc1)(OCC(CF)OC)C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.49
NPC1 O15118 7/20 0.49
SMN1; SMN2 Q16637 6/20 0.49
TP53 P04637 4/20 0.49
MAPT P10636 5/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LMNA P02545 1/20 0.42
GFER P55789 1/20 0.42
KDM4E B2RXH2 2/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20333380 0.75 KMT2A (0.60) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL22216493 0.71 MEN1 (0.60) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL20350547 0.70 ALDH1A1 (0.46) MAPTALDH1A1HSD17B10TDP1LMNA
SCHEMBL29684837 0.70 RAB9A (0.71) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL308069 0.69 NPC1 (0.75) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL22216671 0.69 MEN1 (0.60) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL20347168 0.68 MEN1 (0.56) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL22216571 0.66 ALDH1A1 (0.48) SMN1; SMN2MAPTALDH1A1HSD17B10TDP1
SCHEMBL12495837 0.65 NPC1 (1.00) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL28130084 0.64 RAB9A (1.00) RAB9ANPC1SMN1; SMN2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018119284-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF CALITHERA BIOSCIENCES, INC. (US) 2018-06-28 WO disclosed