SCHEMBL20336147

SCHEMBL20336147

Cc1cc(C2=NCC(c3cc(Cl)cc(Cl)c3)(C(F)(F)F)C2)ccc1C(=O)NCC1CSC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
IKBKB O14920 1/20 0.32
CHRM1 P11229 4/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM3 P20309 1/20 0.32
MAPK14 Q16539 2/20 0.32
CYP3A4 P08684 4/20 0.31
CYP2C9 P11712 4/20 0.31
CYP2C19 P33261 4/20 0.31
CYP2D6 P10635 2/20 0.31
CYP1A2 P05177 2/20 0.31
HDAC4 P56524 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20336185 0.93 NPC1 (0.34) CNR2NPC1RAB9AIKBKBCHRM1
SCHEMBL20336152 0.89 CNR2 (0.34) CNR2CHRM1CHRM2CHRM4CHRM5
SCHEMBL20336181 0.89 CNR2 (0.33) CNR2NPC1RAB9AIKBKBCHRM1
SCHEMBL325802 0.88 TTK (0.34) NPC1RAB9A
SCHEMBL3757227 0.86 ORAI1 (0.33) MAPK14
SCHEMBL20336183 0.86
SCHEMBL14726009 0.84 TTK (0.34) NPC1RAB9A
SCHEMBL14721762 0.83 CNR2 (0.35) CNR2NPC1RAB9ACHRM1CHRM2
SCHEMBL15965601 0.83 CNR2 (0.35) CNR2NPC1RAB9ACHRM1CHRM2
SCHEMBL14721759 0.83 CNR2 (0.35) CNR2NPC1RAB9ACHRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2748154-B1 PROCESS FOR THE PREPARATION OF THIETANE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-07-04 EP disclosed