SCHEMBL20344794

SCHEMBL20344794

CC(=O)c1c(C)cn2cc(-c3cccc(Br)c3)nc2c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.42
SMN1; SMN2 Q16637 7/20 0.42
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
RXFP1 Q9HBX9 1/20 0.42
TP53 P04637 3/20 0.40
ALDH1A1 P00352 6/20 0.40
HCRTR1 O43613 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
POLB P06746 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TSHR P16473 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17029016 0.91 KDM4E (0.45) KDM4ESMN1; SMN2NPC1RAB9ARXFP1
SCHEMBL17029009 0.87 NPC1 (0.43) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL17029025 0.85 KDM4E (0.41) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL18364981 0.81 KMO (0.44) KDM4ESMN1; SMN2NPC1RAB9ARXFP1
SCHEMBL17029008 0.79 KMO (0.43) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL18364982 0.78 RAB9A (0.45) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL17029010 0.77 NPC1 (0.41) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL17029013 0.76 F2RL3 (0.40) KDM4ESMN1; SMN2NPC1RAB9ATP53
SCHEMBL17029007 0.74 XPO1 (0.42) KDM4ESMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL4952276 0.71 CTSS (0.43) KDM4ESMN1; SMN2NPC1RAB9ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2018-07-04 EP disclosed