SCHEMBL20347948

SCHEMBL20347948

Cc1ccc(C(C)(C)C)cc1OCC1CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.45
KDM4E B2RXH2 4/20 0.42
RECQL P46063 1/20 0.40
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP2C9 P11712 1/20 0.38
CNR2 P34972 5/20 0.38
CNR1 P21554 2/20 0.38
EP300 Q09472 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
GRM2 Q14416 1/20 0.36
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
HTR2B P41595 2/20 0.36
GLA P06280 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24334343 0.89 KDM4E (0.54) RIPK1KDM4ERECQLALDH1A1SMN1; SMN2
SCHEMBL14145363 0.86 SCN8A (0.42) RIPK1GRM2
SCHEMBL18120365 0.83 RIPK1 (0.44) RIPK1CNR2CNR1HTR2CHTR2B
SCHEMBL20347946 0.83 DUT (0.46) RIPK1EP300GRM2HTR2AHTR2C
SCHEMBL20347947 0.80 RIPK1 (0.42) RIPK1CNR2CNR1EP300HTR2A
SCHEMBL25510536 0.80 RXRA (0.43) RIPK1ALDH1A1CNR2CNR1EP300
SCHEMBL16662423 0.80 TSHR (0.47) RIPK1KDM4EALDH1A1SMN1; SMN2CYP2C9
SCHEMBL29469863 0.79 RIPK1 (0.44) RIPK1KDM4ERECQLALDH1A1SMN1; SMN2
SCHEMBL24314287 0.79 RIPK1 (0.44) RIPK1KDM4ERECQLALDH1A1SMN1; SMN2
SCHEMBL20206824 0.79 RIPK1 (0.44) RIPK1KDM4EALDH1A1CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230263773-A1 COMBINATION THERAPY WITH DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-08-24 US disclosed
US-20230263773-A1 COMBINATION THERAPY WITH DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-08-24 US disclosed
US-20230126280-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-04-27 US disclosed
US-20230126280-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-04-27 US disclosed
US-11584723-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2023-02-21 US disclosed
US-20220402879-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-12-22 US disclosed
US-11518746-B2 Nitrogen ring linked deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-12-06 US disclosed
US-11247984-B2 Uracil containing compounds CV6 THERAPEUTICS (NI) LIMITED (GB) 2022-02-15 US disclosed
US-11198677-B2 Deoxyuridine triphosphatase inhibitors containing amino sulfonyl linkage UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2021-12-14 US disclosed
US-11174271-B2 6-membered uracil isosteres CV6 THERAPEUTICS (NI) LIMITED (GB) 2021-11-16 US disclosed
US-10562860-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors CV6 THERAPEUTICS (NI) LIMITED (GB) 2020-02-18 US disclosed
US-20200039966-A1 URACIL CONTAINING COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2020-02-06 US disclosed
US-20190276410-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2019-09-12 US disclosed
US-20190270756-A1 6-MEMBERED URACIL ISOSTERES CV6 THERAPEUTICS (NI) LIMITED (GB) 2019-09-05 US disclosed
US-20180201586-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING CYCLOPROPANO LINKAGE SAI LIFE SCIENCES LIMITED (IN) 2018-07-19 US disclosed
US-20180194736-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 US disclosed
US-20180194740-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING AMINO SULFONYL LINKAGE CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 US disclosed
US-20180194740-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING AMINO SULFONYL LINKAGE CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 US disclosed
US-20180186737-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-05 US disclosed
US-20180186737-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (16 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180194736-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885
US-11584723-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885
US-20180194740-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING AMINO SULFONYL LINKAGE DUT, DPYD, TYMP RIPK1 3827/4885KDM4E 1245/4885RECQL 312/4885
US-11174271-B2 6-membered uracil isosteres UNG, DUT, DPYD RIPK1 3321/4885KDM4E 1704/4885RECQL 282/4885
US-20220402879-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885
US-20230263773-A1 COMBINATION THERAPY WITH DEOXYURIDINE TRIPHOSPHATASE INHIBITORS TYMP, DUT, TYMS RIPK1 3821/4885KDM4E 1517/4885RECQL 132/4885
US-20200039966-A1 URACIL CONTAINING COMPOUNDS UNG, DPYD, DUT RIPK1 3431/4885KDM4E 1571/4885RECQL 186/4885
US-11518746-B2 Nitrogen ring linked deoxyuridine triphosphatase inhibitors DUT, DPYD, TYMP RIPK1 3257/4885KDM4E 884/4885RECQL 223/4885
US-11198677-B2 Deoxyuridine triphosphatase inhibitors containing amino sulfonyl linkage DUT, DPYD, TYMP RIPK1 3827/4885KDM4E 1245/4885RECQL 312/4885
US-11247984-B2 Uracil containing compounds UNG, DPYD, DUT RIPK1 3431/4885KDM4E 1571/4885RECQL 186/4885
US-10562860-B2 Hydantoin containing deoxyuridine triphosphatase inhibitors DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885
US-20180186737-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885
US-20190276410-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, DPYD, TYMP RIPK1 3257/4885KDM4E 884/4885RECQL 223/4885
US-20190270756-A1 6-MEMBERED URACIL ISOSTERES UNG, DUT, DPYD RIPK1 3321/4885KDM4E 1704/4885RECQL 282/4885
US-20180201586-A1 DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CONTAINING CYCLOPROPANO LINKAGE DUT, DPYD, TYMP RIPK1 3646/4885KDM4E 1701/4885RECQL 543/4885
US-20230126280-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS DUT, TYMP, DPYD RIPK1 3869/4885KDM4E 1424/4885RECQL 142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.