SCHEMBL20366152

SCHEMBL20366152

COC(=O)[C@H](CCNC(=O)OC(C)(C)C)NC(=O)C[C@@H](C)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GAA P10253 1/20 0.43
TDP1 Q9NUW8 4/20 0.39
ATM Q13315 2/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.37
POLB P06746 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 2/20 0.36
CAPN1 P07384 1/20 0.36
CA14 Q9ULX7 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23685282 0.87 MEN1 (0.43) KLK5MEN1KMT2AGAATDP1
SCHEMBL20366319 0.85 MEN1 (0.47) KLK5MEN1KMT2AGAATDP1
SCHEMBL10164404 0.80 MEN1 (0.47) MEN1KMT2AGAATDP1ATM
SCHEMBL20366165 0.80 MEN1 (0.42) MEN1KMT2AGAATDP1ATM
SCHEMBL20556183 0.79 MEN1 (0.51) MEN1KMT2AGAATDP1ATM
SCHEMBL15159978 0.79 MEN1 (0.51) MEN1KMT2AGAATDP1ATM
SCHEMBL10129167 0.78 MEN1 (0.43) MEN1KMT2AGAATDP1ATM
SCHEMBL11919227 0.77 MEN1 (0.50) KLK5MEN1KMT2AGAATDP1
SCHEMBL21498186 0.77 KMT2A (0.42) KLK5MEN1KMT2AGAATDP1
SCHEMBL5761580 0.76 MEN1 (0.59) MEN1KMT2AGAATDP1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018128826-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF BACTERIAL INFECTIONS CIDARA THERAPEUTICS, INC. (US) 2018-07-12 WO disclosed