SCHEMBL20399604

SCHEMBL20399604

COC(=O)CC1C2CCC1CN(Cc1ccccc1)C2

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.46
S1PR1 P21453 1/20 0.46
S1PR5 Q9H228 1/20 0.46
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29030940 0.86 S1PR1 (0.48) S1PR1S1PR5
SCHEMBL29030939 0.86 S1PR1 (0.48) S1PR1S1PR5
SCHEMBL20399839 0.82 GRIN2B (0.49) GRIN2BS1PR1S1PR5
SCHEMBL6726017 0.80 NR1H2 (0.51) S1PR1S1PR5BCHEACHEMAOB
SCHEMBL26109889 0.79 BCHE (0.52) GRIN2BBCHEACHEMAOB
SCHEMBL8446486 0.78 LTA4H (0.65) BCHEACHEMAOB
SCHEMBL4189224 0.78 GRIN2B (0.48) GRIN2BS1PR1S1PR5
SCHEMBL2980930 0.78 DRD2 (0.67) BCHEACHEMAOB
SCHEMBL4198217 0.76 FUCA1 (0.54) GRIN2BS1PR1S1PR5BCHEACHE
SCHEMBL19971633 0.76 ALDH1A1 (0.53) GRIN2BS1PR1S1PR5BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018136887-A1 COMPOUNDS TESARO, INC. (US) 2018-07-26 WO disclosed