SCHEMBL2040127

SCHEMBL2040127

O=C(O)C1(c2nccs2)CC=CCC1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.35
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2035761 0.82 OPRL1 (0.40) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2037649 0.78 AKR1C1 (0.42) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2035833 0.78 AKR1C1 (0.42) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2035878 0.74 KDM4E (0.35) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2040851 0.70 LMNA (0.39) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL28794538 0.69 OPRL1 (0.34) OPRL1ALDH1A1
SCHEMBL2053963 0.68 LMNA (0.36) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL3797646 0.68 ALDH1A1 (0.35) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2016931 0.67 LMNA (0.38) OPRL1LMNAL3MBTL1ALDH1A1
SCHEMBL2037379 0.66 PDE4A (0.34) OPRL1LMNAL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513098-A1 AMINOPYRIMIDINES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-10-24 EP disclosed
WO-2011075515-A1 AMINOPYRIMIDINES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed