SCHEMBL20405809

SCHEMBL20405809

N/C(=C(\Nc1ccccc1F)c1ccccc1)c1nc(-c2ccc(F)cc2F)no1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
AKR1B1 P15121 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC4 P56524 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RAB9A P51151 6/20 0.36
NPC1 O15118 5/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20406013 0.90 NPC1 (0.43) ALDH1A1LMNAHDAC6RAB9ANPC1
SCHEMBL20405890 0.84 RAB9A (0.45) LMNAHDAC1HDAC4HDAC6RAB9A
SCHEMBL20405898 0.77 ALDH1A1 (0.41) S1PR1ALDH1A1LMNARAB9ANPC1
SCHEMBL20405717 0.76 ALDH1A1 (0.45) ALDH1A1LMNARAB9ANPC1MEN1
SCHEMBL20405797 0.74 ALDH1A1 (0.46) ALDH1A1LMNARAB9ANPC1MEN1
SCHEMBL20405946 0.73 ALDH1A1 (0.42) S1PR1ALDH1A1LMNARAB9ANPC1
SCHEMBL20405810 0.72 ALDH1A1 (0.46) ALDH1A1LMNARAB9ANPC1MEN1
SCHEMBL20405789 0.72 RAB9A (0.42) ALDH1A1LMNAHDAC1HDAC6RAB9A
SCHEMBL2556794 0.70 ALPL (0.50) S1PR1S1PR3AKR1B1HDAC1HDAC4
SCHEMBL20405631 0.70 S1PR1 (0.37) S1PR1S1PR3ALDH1A1LMNAAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250165-B1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO SA (CH) 2018-07-25 EP disclosed