SCHEMBL20439007

SCHEMBL20439007

CC(C)(C)OC(=O)N1CCC(c2c(F)c(F)cc(F)c2F)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.55
KDM4E B2RXH2 1/20 0.55
MAPT P10636 1/20 0.55
DPP4 P27487 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.48
NAMPT P43490 1/20 0.47
GPR119 Q8TDV5 7/20 0.47
TRPV3 Q8NET8 1/20 0.47
TP53 P04637 1/20 0.46
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
PTPN6 P29350 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297784 0.92 KDM4E (0.50) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL28297774 0.92 KDM4E (0.50) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL20439010 0.86 KDM4E (0.55) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL25175456 0.85 THRB (0.54) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL12883601 0.84 GPR119 (0.49) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL12883599 0.84 GPR119 (0.49) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL7982515 0.84 THRB (0.53) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL25939333 0.84 THRB (0.53) THRBKDM4EMAPTDPP4SMN1; SMN2
SCHEMBL28812695 0.83 GPR119 (0.54) THRBKDM4EMAPTSMN1; SMN2NAMPT
SCHEMBL31700475 0.81 MAPT (0.50) THRBKDM4EMAPTDPP4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018137555-A1 POLYFLUORO-SUBSTITUTED AROMATIC HETEROCYCLIC COMPOUND DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND APPLICATIONS THEREOF 浙江大学 2018-08-02 WO disclosed