SCHEMBL20439234

SCHEMBL20439234

CNC(=O)c1cc(Oc2ccccc2)ccc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.56
HDAC8 Q9BY41 6/20 0.55
BRAF P15056 6/20 0.55
HDAC1 Q13547 6/20 0.55
HDAC3 O15379 5/20 0.55
HDAC4 P56524 5/20 0.55
HDAC7 Q8WUI4 5/20 0.55
HDAC2 Q92769 5/20 0.55
HDAC10 Q969S8 5/20 0.55
HDAC11 Q96DB2 5/20 0.55
HDAC6 Q9UBN7 5/20 0.55
HDAC9 Q9UKV0 5/20 0.55
HDAC5 Q9UQL6 5/20 0.55
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
GCK P35557 2/20 0.49
MMP13 P45452 1/20 0.49
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31557926 0.86 BRAF (0.61) HDAC8BRAFHDAC1HDAC3HDAC4
SCHEMBL20439216 0.84 HPGD (0.61) HPGDHTTSMN1; SMN2MMP13LMNA
SCHEMBL13714246 0.83 NR1H4 (0.65) NR1H4MAPK1GFERTDP1SRD5A2
SCHEMBL15028056 0.83 NR1H4 (0.53) NR1H4HPGDSMN1; SMN2MAPK1GFER
SCHEMBL23052920 0.82 NR1H4 (0.56) NR1H4HPGDSMN1; SMN2MAPK1GFER
SCHEMBL31557904 0.81 MEN1 (0.50) HDAC8BRAFHDAC1HDAC3HDAC4
SCHEMBL8360010 0.80 MTNR1A (0.56) BRAFHDAC1HPGDHTTLMNA
Hydrochloric Acid SCHEMBL27696847 0.79 PARP10 (0.54) NR1H4GCKSRD5A2CYP1A2CYP2C9
SCHEMBL28173271 0.78 BRAF (0.49) HDAC8BRAFHDAC1HDAC3HDAC4
SCHEMBL31557917 0.76 BRAF (0.44) NR1H4HDAC8BRAFHDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018140186-A1 A PROCESS FOR PREPARING 5-PHENOXY-1(3H)ISOBENZOFURANONE KINGCHEM LIFE SCIENCE LLC (US) 2018-08-02 WO disclosed