SCHEMBL8360010

SCHEMBL8360010

CNC(=O)c1cc(OC)ccc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.56
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 4/20 0.55
GAA P10253 3/20 0.55
HPGD P15428 3/20 0.55
HSD17B10 Q99714 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CASP1 P29466 1/20 0.55
CASP7 P55210 1/20 0.55
PLK1 P53350 1/20 0.55
GLA P06280 1/20 0.52
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HTT P42858 2/20 0.49
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HSD17B1 P14061 2/20 0.47
HSD17B2 P37059 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767061 0.86 PLK1 (0.59) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL17414607 0.82 P2RX1 (0.57) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL29502160 0.81 KDM4E (0.62) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL146258 0.81 KDM4E (0.62) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL1558756 0.81 BRAF (0.65) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL7502111 0.81 HPGD (0.61) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL18661182 0.81 MTNR1A (0.55) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL7984549 0.81 TYK2 (0.62) MTNR1AALDH1A1KDM4EGAAHPGD
SCHEMBL20439234 0.80 NR1H4 (0.56) HPGDHTTCYP2C9CYP1A2RAF1
SCHEMBL1986986 0.79 ALDH1A1 (0.61) ALDH1A1KDM4EGAAHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003026652-A1 LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-04-03 WO disclosed
US-4107311-A ANTI-FERTILITY AGENTS, ABORTIFACIENTS SANDOZ, INC. (US) 1978-08-15 US disclosed