SCHEMBL20439372

SCHEMBL20439372

Oc1c(Br)ccc2[nH]ncc12

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 6/20 0.55
AXL P30530 2/20 0.55
IDO1 P14902 7/20 0.43
TDO2 P48775 3/20 0.43
METAP2 P50579 3/20 0.41
CSNK2A1 P68400 1/20 0.41
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
DYRK1A Q13627 1/20 0.37
PTPN6 P29350 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21437262 0.79 NOS1 (0.44) NOS1AXLIDO1METAP2CCNA2
SCHEMBL767109 0.76 NOS1 (0.55) NOS1AXLIDO1TDO2METAP2
SCHEMBL12821601 0.76 NOS1 (0.55) NOS1AXLIDO1TDO2METAP2
SCHEMBL767506 0.76 NOS1 (0.55) NOS1AXLIDO1TDO2METAP2
SCHEMBL5413400 0.76 NOS1 (0.50) NOS1AXLIDO1TDO2METAP2
SCHEMBL767674 0.76 NOS1 (0.55) NOS1AXLIDO1TDO2METAP2
SCHEMBL12321248 0.75 NOS1 (0.56) NOS1AXLIDO1TDO2METAP2
SCHEMBL6923181 0.74 NOS1 (0.49) NOS1AXLIDO1TDO2METAP2
SCHEMBL21196087 0.72 TRPA1 (0.41) NOS1AXLIDO1CCNA2CDK2
SCHEMBL1141845 0.72 NOS1 (0.50) NOS1AXLIDO1TDO2METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018138739-A1 NOVEL ANTIESTROGENIC HETEROCYCLIC COMPOUNDS SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED (IN) 2018-08-02 WO disclosed