SCHEMBL20439386

SCHEMBL20439386

CNC(COc1cc(OCc2ccccc2)ccc1Br)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 1/20 0.40
RECQL P46063 1/20 0.40
HTR1D P28221 2/20 0.39
GPR34 Q9UPC5 2/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
FFAR1 O14842 2/20 0.38
AR P10275 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PTPN1 P18031 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20439317 0.90 MAOB (0.38) MAOBALDH1A1HTR1D
SCHEMBL20439308 0.83 MAOB (0.44) MAOBKMT2AMEN1ALDH1A1RECQL
SCHEMBL20439307 0.83 MAOB (0.44) MAOBKMT2AMEN1ALDH1A1RECQL
SCHEMBL20439384 0.83 PTPN1 (0.43) KMT2AMEN1ALDH1A1GPR34FFAR1
SCHEMBL20439374 0.79 LMNA (0.40) KMT2AMEN1ALDH1A1HTR1DFFAR1
SCHEMBL5354486 0.76 BCL2 (0.44) PTPN1
SCHEMBL20439435 0.76 BCL2 (0.44) PTPN1
SCHEMBL20425144 0.76 MAOB (0.43) MAOBKMT2AMEN1ALDH1A1RECQL
SCHEMBL5355437 0.76 SCN4A (0.48) MAOBKMT2ALMNAMAPT
SCHEMBL20439319 0.76 SCN4A (0.48) MAOBKMT2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018138739-A1 NOVEL ANTIESTROGENIC HETEROCYCLIC COMPOUNDS SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED (IN) 2018-08-02 WO disclosed