SCHEMBL20439384

SCHEMBL20439384

CC(C)(C)OC(=O)N[C@@H](COc1cc(OCc2ccccc2)ccc1Br)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.43
GPR34 Q9UPC5 2/20 0.41
PPARA Q07869 1/20 0.41
BCL2 P10415 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
CTSS P25774 2/20 0.39
FFAR1 O14842 2/20 0.39
FFAR4 Q5NUL3 1/20 0.39
PRKCA P17252 1/20 0.39
PRKCD Q05655 1/20 0.39
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
JAK2 O60674 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354486 0.94 BCL2 (0.44) PTPN1PPARABCL2CTSSPRKCA
SCHEMBL20439435 0.94 BCL2 (0.44) PTPN1PPARABCL2CTSSPRKCA
SCHEMBL20439315 0.92 PTPN1 (0.41) PTPN1PPARABCL2AAK1CTSS
SCHEMBL20439373 0.83 AAK1 (0.43) PPARAAAK1ALDH1A1HTTNPSR1
SCHEMBL20439398 0.83 AAK1 (0.43) PPARAAAK1ALDH1A1HTTNPSR1
SCHEMBL20439386 0.83 MAOB (0.41) PTPN1GPR34FFAR1FFAR4MEN1
SCHEMBL20439399 0.78 BCL2 (0.43) PTPN1PPARABCL2PRKCAPRKCD
SCHEMBL20439397 0.78 BCL2 (0.43) PTPN1PPARABCL2PRKCAPRKCD
SCHEMBL5350616 0.76 PRKCA (0.54) PTPN1PPARABCL2PRKCAPRKCD
SCHEMBL1553475 0.76 PRKCA (0.54) PTPN1PPARABCL2PRKCAPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018138739-A1 NOVEL ANTIESTROGENIC HETEROCYCLIC COMPOUNDS SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED (IN) 2018-08-02 WO disclosed