SCHEMBL20442602

SCHEMBL20442602

CCOc1ccc(OCCBr)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.67
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
TDP1 Q9NUW8 2/20 0.54
TSHR P16473 1/20 0.54
LTA4H P09960 2/20 0.50
RECQL P46063 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
PARP10 Q53GL7 1/20 0.45
RELA Q04206 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
PRSS1 P07477 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8140756 0.87 NPC1 (0.47) NQO1ALDH1A1SMN1; SMN2LTA4HRECQL
SCHEMBL13303281 0.86 LTA4H (0.57) TSHRLTA4HCYP1A2CYP2D6CYP2C19
SCHEMBL5726997 0.83 MAPK1 (0.56) NQO1KDM4EALDH1A1TDP1TSHR
SCHEMBL2412878 0.82 LMNA (0.55) KDM4EALDH1A1SMN1; SMN2TDP1LTA4H
1,4-Diethoxybenzene SCHEMBL124015 0.82 NQO1 (1.00) NQO1KDM4EALDH1A1SMN1; SMN2TDP1
1,4-Diethoxybenzene SCHEMBL28186701 0.82 NQO1 (1.00) NQO1KDM4EALDH1A1SMN1; SMN2TDP1
SCHEMBL896082 0.81 CA12 (0.52) KDM4EALDH1A1SMN1; SMN2TDP1L3MBTL1
SCHEMBL2414381 0.81 DRD2 (0.55) KDM4EALDH1A1SMN1; SMN2L3MBTL1
4-Ethoxy-1-Propoxybenzene SCHEMBL2841577 0.80 NQO1 (0.74) NQO1KDM4EALDH1A1SMN1; SMN2TDP1
SCHEMBL14984021 0.80 NQO1 (0.74) NQO1KDM4EALDH1A1SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018140809-A1 MODULATORS OF ESTROGEN RECEPTOR PROTEOLYSIS AND ASSOCIATED METHODS OF USE Arvinas, Inc. (US) 2018-08-02 WO disclosed