SCHEMBL20443196

SCHEMBL20443196

CC(C)(C(F)(F)F)S(=O)(=O)c1ccc(F)c(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 11/20 0.45
IDO1 P14902 1/20 0.38
CA2 P00918 5/20 0.38
CA1 P00915 4/20 0.38
CA9 Q16790 1/20 0.35
ALDH1A1 P00352 1/20 0.35
VCP P55072 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15068050 0.82 EPAS1 (0.60) EPAS1CA2ALDH1A1
SCHEMBL23358269 0.78 CNR2 (0.42) EPAS1IDO1CA2CA1CA9
SCHEMBL29887062 0.74 EPAS1 (0.51) EPAS1IDO1CA2CA1CA9
SCHEMBL2381326 0.74 EPAS1 (0.51) EPAS1IDO1CA2CA1CA9
SCHEMBL29555632 0.74 VCAM1 (0.52) EPAS1IDO1CA2CA1CA9
SCHEMBL5150927 0.74 VCAM1 (0.52) EPAS1IDO1CA2CA1CA9
SCHEMBL21190881 0.73 KMT2A (0.51) IDO1ALDH1A1
Ethane SCHEMBL26669304 0.73 CA2 (0.57) CA2CA1CA9
SCHEMBL15068035 0.72 CA2 (0.61) CA2CA1CA9
SCHEMBL20384341 0.72 EPAS1 (0.43) EPAS1IDO1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110198941-B Pyrrolopyridine N-oxide derivative and preparation method and application thereof 江苏豪森药业集团有限公司 2021-09-28 CN disclosed
WO-2018137655-A1 PYRROLO-PYRIDINES N-OXIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-08-02 WO disclosed