SCHEMBL20458161

SCHEMBL20458161

O=C(O)C1CCN1c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.53
ALOX12 P18054 2/20 0.47
THRB P10828 1/20 0.47
KMT2A Q03164 1/20 0.47
MAPT P10636 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 2/20 0.41
MAPK1 P28482 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9891645 1.00 NOTUM (0.53) NOTUMALOX12THRBKMT2AMAPT
SCHEMBL5702089 0.83 NOTUM (0.49) NOTUMKMT2AALDH1A1SMN1; SMN2
SCHEMBL5702158 0.83 NOTUM (0.49) NOTUMKMT2AALDH1A1SMN1; SMN2
SCHEMBL13015198 0.82 GFER (0.41) NOTUMALOX12THRBKMT2AMAPT
SCHEMBL2121764 0.82 NOTUM (0.53) NOTUMKMT2AMAPTALDH1A1HPGD
SCHEMBL2121761 0.82 NOTUM (0.53) NOTUMKMT2AMAPTALDH1A1HPGD
SCHEMBL7035832 0.82 GFER (0.41) NOTUMALOX12THRBKMT2AMAPT
SCHEMBL21660768 0.80 SCN9A (0.43) NOTUMKMT2AHRH3CA1CA2
SCHEMBL20141514 0.80 NOTUM (0.48) NOTUMALOX12THRBKMT2AMAPT
SCHEMBL5394683 0.79 NOTUM (0.43) NOTUMALOX12THRBKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443107-B1 AZETIDINE 2 -CARBOXAMIDE DERIVATIVES WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INT (DE) 2018-08-08 EP disclosed