SCHEMBL20469120

SCHEMBL20469120

Cc1ccc(C#Cc2ccc(N3C[C@@H](C)O[C@@H](C)C3)nc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.51
MTOR P42345 1/20 0.51
GRM5 P41594 7/20 0.47
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
AOC3 Q16853 1/20 0.41
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24018507 0.84 KMT2A (0.53) KMT2AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL31182223 0.84 KMT2A (0.53) KMT2AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL18436130 0.84 KMT2A (0.53) KMT2AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL15743968 0.84 KMT2A (0.53) KMT2AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL10034110 0.84 KMT2A (0.53) KMT2AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL20456767 0.81 KMT2A (0.48) PIK3CAMTORGRM5KMT2AALDH1A1
SCHEMBL20469115 0.80 CHRNB2 (0.43) GRM5
SCHEMBL20468981 0.77 GRM5 (0.39) GRM5
SCHEMBL23253135 0.77 PIK3CA (0.54) PIK3CAMTORGRM5ALDH1A1LMNA
SCHEMBL20469234 0.74 GRM5 (0.42) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3909949-A1 ATAZANAVIR (ATV) ANALOGUES FOR TREATING HIV INFECTIONS Gilead Sciences, Inc. (US) 2021-11-17 EP disclosed
EP-3577110-B1 8-OXETAN-3-YL-3,8-DIAZABICYCLO[3.2.1]OCTAN-3-YL SUBSTITUTED COMPOUNDS AS HIV INHIBITORS GILEAD SCIENCES INC (US) 2021-04-21 EP disclosed
WO-2018145021-A1 ATAZANAVIR (ATV) ANALOGUES FOR TREATING HIV INFECTIONS GILEAD SCIENCES, INC. (US) 2018-08-09 WO disclosed