SCHEMBL20470544

SCHEMBL20470544

C#Cc1cc(CC)ccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.41
PYCR1 P32322 2/20 0.37
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RXRG P48443 2/20 0.35
AR P10275 4/20 0.35
TRPA1 O75762 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
CYP2A6 P11509 2/20 0.33
KIF11 P52732 1/20 0.33
CYP1A2 P05177 1/20 0.33
PDK2 Q15119 1/20 0.33
HSD11B1 P28845 1/20 0.33
FFAR1 O14842 1/20 0.33
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16691050 0.82 AR (0.48) RXRARXRBRXRGARCYP2A6
SCHEMBL3245823 0.81 RXRA (0.44) PDE2APYCR1RXRARXRBRXRG
SCHEMBL25909005 0.79 RXRA (0.39) PYCR1RXRARXRBRXRGAR
SCHEMBL8196522 0.76 TRPA1 (0.38) PYCR1TRPA1CYP2A6KIF11CYP1A2
SCHEMBL20455595 0.76 AR (0.42) PDE2AARKIF11HSD11B1
SCHEMBL29890778 0.76 AR (0.42) PDE2AARKIF11HSD11B1
SCHEMBL12706035 0.73 KIF11 (0.53) TRPA1KIF11FFAR1DAO
SCHEMBL26145454 0.73 FFAR4 (0.40) PDE2ARXRARXRBRXRGAR
SCHEMBL12886693 0.73 PDE2A (0.53) PDE2ARXRARXRBRXRGTRPA1
SCHEMBL29892139 0.73 IDO1 (0.38) ARTRPA1KIF11HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018141857-A1 ARYL HYDROCARBON RECEPTOR (AHR) MODULATOR COMPOUNDS PHENEX PHARMACEUTICALS AG (DE) 2018-08-09 WO disclosed