SCHEMBL2050249

SCHEMBL2050249

C=CCC1CCC(CO)CC1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.34
ESR2 Q92731 6/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
TSHR P16473 1/20 0.33
NOS3 P29474 2/20 0.31
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678892 1.00 ESR1 (0.34) ESR1ESR2CYP3A4CYP2C9TSHR
SCHEMBL6683176 0.93 ESR1 (0.31) ESR1ESR2CYP3A4CYP2C9
SCHEMBL6683178 0.93 ESR1 (0.31) ESR1ESR2CYP3A4CYP2C9
SCHEMBL432351 0.86
SCHEMBL815076 0.86 NOS1 (0.37) NOS3NOS1NOS2
SCHEMBL5888802 0.85 EPHX2 (0.31) TSHR
SCHEMBL15536154 0.83
Butadiene SCHEMBL3476348 0.80 ESR1 (0.38) ESR1ESR2CYP3A4CYP2C9TSHR
SCHEMBL9556372 0.80 ESR2 (0.38) ESR2TSHR
SCHEMBL9556377 0.80 ESR2 (0.38) ESR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2247146-A None JP disclosed
JP-7313177-A None JP disclosed
JP-63006056-A None JP disclosed
US-20110141418-A1 LIQUID CRYSTAL COMPOUNDS QINETIQ LIMITED (GB) 2011-06-16 US disclosed
EP-1905597-B1 Inkjet recording apparatus FUJIFILM CORP (JP) 2010-11-03 EP disclosed
US-7671191-B2 Methods for preparing 2-alkynyladenosine derivatives PGX HEALTH, LLC (US) 2010-03-02 US disclosed
US-20080177055-A1 Methods for preparing 2-alkynyladenosine deriviatives ADENOSINE THERAPEUTICS, LLC 2008-07-24 US disclosed
EP-1905597-A2 Inkjet recording apparatus FUJIFILM Corporation (JP) 2008-04-02 EP disclosed
JP-H07313177-A PRODUCTION OF TRANS-CYCLOHEXYLMETHYL ESTER ASAHI DENKA KOGYO KK 1995-12-05 JP disclosed
US-5354502-A Very large dielectric anisotropy and small birefringence SEIKO EPSON CORPORATION (JP) 1994-10-11 US disclosed
US-5238599-A Low threshold voltage, low driving voltage SEIKO EPSON CORPORATION (JP) 1993-08-24 US disclosed
EP-0447565-A1 1,3-DIOXANE DERIVATIVE AND LIQUID-CRYSTAL COMPOSITION CONTAINING THE SAME SEIKO EPSON CORPORATION (JP) 1991-09-25 EP disclosed
EP-0400861-A1 1,3-dioxane derivative and liquid crystal composition incorporating the same SEIKO EPSON CORPORATION (JP) 1990-12-05 EP disclosed
JP-H02247146-A TRICYCLIC COMPOUND HAVING OXYMETHYLENE BOND DAINIPPON INK & CHEM INC 1990-10-02 JP disclosed
JP-S636056-A ANTHRAQUINONE DYE AND LIQUID CRYSTAL COMPOSITION CONTAINING SAME NIPPON KANKO SHIKISO KENKYUSHO:KK 1988-01-12 JP disclosed
EP-0058512-B1 LIQUID CRYSTAL COMPOUNDS EXHIBITING A SMALL DIELECTRIC ANISOTROPY AND LIQUID CRYSTAL MATERIALS AND DEVICES INCORPORATING SUCH COMPOUNDS The Secretary of State for Defence in Her Britannic Majesty's Government of the United Kingdom of Great Britain and (GB) 1986-01-15 EP disclosed
US-4556745-A BICYCOL(2.2.2) OCATANE RING THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 1985-12-03 US disclosed
US-4357078-A ELECTROOPTICS; DISPLAYING THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 1982-11-02 US disclosed
EP-0058512-A1 Liquid crystal compounds exhibiting a small dielectric anisotropy and liquid crystal materials and devices incorporating such compounds The Secretary of State for Defence in Her Britannic Majesty's Government of the United Kingdom of Great Britain and (GB) 1982-08-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110141418-A1 LIQUID CRYSTAL COMPOUNDS HTR3D, HTR3C, SFXN3 ESR1 4503/4885ESR2 4461/4885CYP3A4 2396/4885
US-20080177055-A1 Methods for preparing 2-alkynyladenosine deriviatives ADORA2A, ADORA3, ADORA1 ESR1 3087/4885ESR2 2823/4885CYP3A4 2261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.