SCHEMBL2051091

SCHEMBL2051091

Fc1cccc(-c2cc[c]c(C(F)(F)F)c2)c1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
PGR P06401 2/20 0.35
TRPA1 O75762 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
DYRK1A Q13627 2/20 0.32
PLK4 O00444 1/20 0.32
MAPK13 O15264 1/20 0.32
DAPK3 O43293 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
CDK1 P06493 1/20 0.32
PIM1 P11309 1/20 0.32
CDK2 P24941 1/20 0.32
MARK3 P27448 1/20 0.32
FLT4 P35916 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
CDK8 P49336 1/20 0.32
CLK2 P49760 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2431244 0.87 PDK2 (0.42) PGRTRPA1MAP4K4PDK2BACE1
SCHEMBL15638417 0.84 AR (0.38) PDK2CHRM5GPBAR1
SCHEMBL2053032 0.81 TRPA1 (0.38) TRPA1PDK2
SCHEMBL15637692 0.81 GABRA1 (0.40) PGR
SCHEMBL8115423 0.80 PGR (0.38) PGRPDE3BPDE3ADYRK1APLK4
SCHEMBL15637441 0.78 ESR1 (0.30)
SCHEMBL11131265 0.77 PDK2 (0.35) TRPA1PDE3BPDE3APDK2BACE1
SCHEMBL2014094 0.77 PGR (0.39) HSD11B1PGRDYRK1APLK4MAPK13
SCHEMBL6668303 0.77 AR (0.51) HSD11B1PGRTRPA1CLK4BACE1
SCHEMBL15636571 0.77 PGR (0.36) PGRDYRK1APLK4MAPK13DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed