SCHEMBL20535503

SCHEMBL20535503

C[Si](C)(C)CCOCn1ccc2c(Cl)cc(Br)cc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 4/20 0.36
NPC1 O15118 1/20 0.33
EGFR P00533 1/20 0.31
IGF1R P08069 1/20 0.31
SRC P12931 1/20 0.31
FLT4 P35916 1/20 0.31
KDR P35968 1/20 0.31
FLT3 P36888 1/20 0.31
EPHB4 P54760 1/20 0.31
TEK Q02763 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23326408 0.82 NPC1 (0.36) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL19252060 0.82 DGAT1 (0.36) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL30930962 0.82 DGAT1 (0.36) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL29910227 0.81 DGAT1 (0.36) DGAT1NPC1
SCHEMBL23326567 0.81 DGAT1 (0.36) DGAT1NPC1
SCHEMBL23326337 0.81 DGAT1 (0.34) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL20535513 0.79 RHEB (0.36) NPC1MAPT
SCHEMBL16076726 0.79 NPC1 (0.36) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL18321909 0.78 DGAT1 (0.35) DGAT1NPC1EGFRIGF1RSRC
SCHEMBL30475587 0.77 HTR7 (0.42) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11339144-B2 Heteroaryl Rheb inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2022-05-24 US disclosed
US-20210238165-A1 HETEROARYL RHEB INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2021-08-05 US disclosed
WO-2018191146-A1 HETEROARYL RHEB INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210238165-A1 HETEROARYL RHEB INHIBITORS AND USES THEREOF RHEB, KRAS, NRAS DGAT1 3962/4885NPC1 868/4885EGFR 1990/4885
US-11339144-B2 Heteroaryl Rheb inhibitors and uses thereof RHEB, GDI2, KRAS DGAT1 2656/4885NPC1 403/4885EGFR 2403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.