Bromide

Bromide

SCHEMBL20536256

Br.N#Cc1cnc([Zn])cc1-c1ccccc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
NPSR1 Q6W5P4 3/20 0.51
TDP1 Q9NUW8 3/20 0.51
KDM4E B2RXH2 5/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
CYP1A2 P05177 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 3/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
CYP19A1 P11511 2/20 0.43
LRRK2 Q5S007 3/20 0.42
KDR P35968 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7213782 0.84 NPSR1 (0.53) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL14379730 0.81 ALDH1A1 (0.50) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL14379734 0.81 ALDH1A1 (0.50) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
Bromide SCHEMBL20536252 0.79 ALDH1A1 (0.49) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL20536253 0.78 ALDH1A1 (0.47) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL25204363 0.77 NPSR1 (0.46) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL29466494 0.74 ALDH1A1 (0.49) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
Bromide SCHEMBL20536675 0.74 RPS6KA3 (0.39) ADORA1NPC1RAB9A
SCHEMBL30603820 0.72 PDPK1 (0.50) ALDH1A1NPSR1TDP1KDM4EL3MBTL1
SCHEMBL30603821 0.72 HPGDS (0.50) ALDH1A1NPSR1TDP1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10937974-B2 Organometallic compound, organic light-emitting device including the organometallic compound, and diagnostic composition including the organometallic compound SAMSUNG ELECTRONICS CO; LTD. (KR) 2021-03-02 US disclosed
EP-3392257-B1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE ORGANOMETALLIC COMPOUND, AND DIAGNOSTIC COMPOSITION INCLUDING THE ORGANOMETALLIC COMPOUND SAMSUNG ELECTRONICS CO LTD (KR) 2020-06-10 EP disclosed
US-20180309071-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE ORGANOMETALLIC COMPOUND, AND DIAGNOSTIC COMPOSITION INCLUDING THE ORGANOMETALLIC COMPOUND SAMSUNG ELECTRONICS CO., LTD. (KR) 2018-10-25 US disclosed
EP-3392257-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE ORGANOMETALLIC COMPOUND, AND DIAGNOSTIC COMPOSITION INCLUDING THE ORGANOMETALLIC COMPOUND Samsung Electronics Co., Ltd. (KR) 2018-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180309071-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE ORGANOMETALLIC COMPOUND, AND DIAGNOSTIC COMPOSITION INCLUDING THE ORGANOMETALLIC COMPOUND ORC3, LEF1, OCIAD1 ALDH1A1 147/4885NPSR1 4827/4885TDP1 3297/4885
US-10937974-B2 Organometallic compound, organic light-emitting device including the organometallic compound, and diagnostic composition including the organometallic compound ORC3, LEF1, OCIAD1 ALDH1A1 147/4885NPSR1 4827/4885TDP1 3297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.