SCHEMBL2056440

SCHEMBL2056440

CCCCOc1nc(N)nc2[nH]c(CCCNC(=O)OC(C)(C)C)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.43
CA2 P00918 6/20 0.43
CA12 O43570 5/20 0.43
CA9 Q16790 5/20 0.43
TLR7 Q9NYK1 7/20 0.39
IL6 P05231 2/20 0.37
STK17B O94768 1/20 0.37
STK17A Q9UEE5 1/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
PIN1 Q13526 1/20 0.35
BCHE P06276 1/20 0.35
CACNA1H O95180 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054844 0.85 L3MBTL1 (0.43) CA1CA2CA12CA9TLR7
SCHEMBL2097032 0.84 CA1 (0.39) CA1CA2CA12CA9TLR7
SCHEMBL2054806 0.83 STK17B (0.42) CA1CA2CA12CA9STK17B
SCHEMBL2054842 0.80 PIN1 (0.51) CA1CA2CA12CA9MEN1
SCHEMBL14404995 0.80 TDP1 (0.38) CA1CA2CA12CA9STK17B
SCHEMBL2054792 0.77 CACNA1H (0.35) CA1CA2CA12CA9STK17B
SCHEMBL2054834 0.76 TDP1 (0.40) CA1CA2CA12CA9STK17B
SCHEMBL2056437 0.70 CA1 (0.43) CA1CA2CA12CA9TLR7
SCHEMBL6004545 0.68 NPSR1 (0.44) CA1CA2CA12CA9TLR7
SCHEMBL6007018 0.68 NPSR1 (0.44) CA1CA2CA12CA9TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730298-B1 SPECIFIC SUBSTRATES FOR O6-ALKYLGUANINE-DNA ALKYLTRANSFERASE EPFL ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (CH) 2015-11-11 EP disclosed
US-8163479-B2 Specific substrates for O6-alkylguanine-DNA alkyltransferase ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2012-04-24 US disclosed
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase EPFL ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (CH) 2007-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070243568-A1 Specific Substrates for O6-Alkylguanine-Dna Alkyltransferase AGT, AGXT, AGTR1 CA1 4500/4885CA2 3221/4885CA12 4578/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.