SCHEMBL20569138

SCHEMBL20569138

COC(=O)c1cccc(Cn2ccnc2C(C)O)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.53
OPRD1 P41143 1/20 0.52
LOXL2 Q9Y4K0 1/20 0.48
YTHDC1 Q96MU7 1/20 0.48
CYP4F2 P78329 2/20 0.47
CYP4A11 Q02928 2/20 0.47
ABHD6 Q9BV23 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
SLC7A5 Q01650 1/20 0.45
CD74 P04233 1/20 0.45
MIF P14174 1/20 0.45
MAPK10 P53779 1/20 0.45
KDM4E B2RXH2 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20570142 0.87 HTT (0.52) IDO1YTHDC1TDP1KMT2ACYP1A2
SCHEMBL20569345 0.84 BRD4 (0.44) TDP1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL20570136 0.79 TSHR (0.53) TDP1KMT2ACYP1A2CYP2D6CYP2C19
Iodide SCHEMBL29037976 0.76 TDP1 (0.61) TDP1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL696380 0.74 OPRD1 (0.52) IDO1OPRD1LOXL2YTHDC1CYP4F2
SCHEMBL7830882 0.73 LOXL2 (0.62) IDO1LOXL2CYP4F2CYP4A11ABHD6
SCHEMBL696367 0.73 OPRD1 (0.51) IDO1OPRD1LOXL2YTHDC1KMT2A
SCHEMBL14987126 0.73 HTT (0.71) IDO1LOXL2CYP4F2CYP4A11ABHD6
SCHEMBL20570065 0.73 CYP1A2 (0.48) TDP1KMT2ACYP1A2CYP2D6CYP2C19
SCHEMBL697926 0.73 RAB9A (0.48) OPRD1YTHDC1TDP1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018216822-A1 NOVEL IMIDAZOLE DERIVATIVES TAISHO PHARMACEUTICAL CO., LTD. (JP) 2018-11-29 WO disclosed