SCHEMBL20569640

SCHEMBL20569640

CN(C)CCn1c(=O)n(CCC(C)(C)O)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.51
CNR1 P21554 1/20 0.49
POLB P06746 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP1A2 P05177 1/20 0.44
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
TOP2A P11388 1/20 0.42
HDAC1 Q13547 1/20 0.40
APEX1 P27695 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR6 P50406 2/20 0.39
SIGMAR1 Q99720 1/20 0.38
MPO P05164 1/20 0.38
HAVCR2 Q8TDQ0 1/20 0.38
CYP2D6 P10635 1/20 0.38
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745333 0.89 CNR2 (0.56) CNR2CNR1ALDH1A1CYP1A2NPC1
SCHEMBL31357282 0.83 CNR2 (0.52) CNR2CNR1ALDH1A1NPC1GAA
SCHEMBL30904706 0.81 CNR1 (0.53) CNR2CNR1POLBALDH1A1CYP1A2
SCHEMBL13354930 0.78 CYP1A2 (0.56) CNR2POLBALDH1A1CYP1A2NPC1
SCHEMBL12933336 0.73 TOP2A (0.51) CNR2ALDH1A1TOP2AHDAC1HTR6
SCHEMBL13322672 0.73 CNR2 (0.47) CNR2POLBALDH1A1CYP1A2TOP2A
SCHEMBL22700957 0.73 NPC1 (0.47) CNR2CNR1ALDH1A1CYP1A2NPC1
SCHEMBL20569856 0.72 KDM4E (0.58) CNR2CNR1ALDH1A1GAA
SCHEMBL1128490 0.71 FABP4 (0.50) CNR2CNR1ALDH1A1CYP1A2HDAC1
SCHEMBL8347752 0.71 MAPK8 (0.55) CNR2ALDH1A1TOP2AHDAC1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3630291-A1 BENZIMIDAZOLONE DERIVED INHIBITORS OF BCL6 Cancer Research Technology Limited (GB) 2020-04-08 EP claimed
WO-2018215801-A1 BENZIMIDAZOLONE DERIVED INHIBITORS OF BCL6 CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-11-29 WO claimed