SCHEMBL20576367

SCHEMBL20576367

Fc1ccccc1-c1cc(Cl)nc(Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
HSP90AA1 P07900 2/20 0.46
HSP90AB1 P08238 2/20 0.46
MPL P40238 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADORA2A P29274 5/20 0.41
ADORA1 P30542 4/20 0.41
ADORA3 P0DMS8 3/20 0.41
ADORA2B P29275 1/20 0.41
IDO1 P14902 1/20 0.41
KDM5B Q9UGL1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20910316 0.90 L3MBTL1 (0.52) NPC1L3MBTL1CASP3SENP8SENP7
SCHEMBL29502717 0.82 HSP90AA1 (0.70) NPC1HSP90AA1HSP90AB1MPLADORA2A
SCHEMBL17476767 0.82 HSP90AA1 (0.70) NPC1HSP90AA1HSP90AB1MPLADORA2A
SCHEMBL602995 0.82 MAPK14 (0.45) NPC1L3MBTL1CASP3SENP8SENP7
SCHEMBL3327517 0.81 HSP90AA1 (0.68) NPC1L3MBTL1HSP90AA1HSP90AB1MEN1
SCHEMBL22084208 0.78 ALDH1A1 (0.57) L3MBTL1HSP90AA1HSP90AB1MEN1ALDH1A1
SCHEMBL21058449 0.78 HSP90AA1 (0.46) NPC1L3MBTL1CASP3SENP8SENP7
SCHEMBL21058751 0.77 ACP1 (0.47) L3MBTL1HSP90AA1HSP90AB1MEN1ALDH1A1
SCHEMBL12579954 0.76 HSP90AA1 (0.49) L3MBTL1HSP90AA1HSP90AB1MEN1ALDH1A1
SCHEMBL786422 0.76 HSD11B1 (0.41) NPC1HSP90AA1HSP90AB1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3362451-B1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2023-04-12 EP disclosed
US-11225477-B2 Inhibitors of influenza virus replication, application methods and uses thereof SUNSHINE LAKE PHARMA CO., LTD. (CN) 2022-01-18 US disclosed
US-20200299294-A1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2020-09-24 US disclosed
US-10717732-B2 Inhibitors of influenza virus replication, application methods and uses thereof SUNSHINE LAKE PHARMA CO., LTD. (CN) 2020-07-21 US disclosed
CN-106854205-B Inhibitors of influenza virus replication and methods of use and uses thereof 广东东阳光药业有限公司 2019-07-09 CN disclosed
CN-109748915-A Inhibitors of influenza viruses replication and its application method and purposes 广东东阳光药业有限公司 2019-05-14 CN disclosed
US-20180346463-A1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2018-12-06 US disclosed
CN-106854205-A Inhibitors of influenza virus replication and methods of use and uses thereof 广东东阳光药业有限公司 2017-06-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200299294-A1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF POLRMT, EIF2AK2, POLM NPC1 2126/4885L3MBTL1 3838/4885CASP3 4330/4885
US-20180346463-A1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF POLRMT, EIF2AK2, POLM NPC1 2126/4885L3MBTL1 3838/4885CASP3 4330/4885
US-10717732-B2 Inhibitors of influenza virus replication, application methods and uses thereof POLRMT, EIF2AK2, POLM NPC1 2126/4885L3MBTL1 3838/4885CASP3 4330/4885
US-11225477-B2 Inhibitors of influenza virus replication, application methods and uses thereof POLRMT, EIF2AK2, POLM NPC1 2126/4885L3MBTL1 3838/4885CASP3 4330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.