SCHEMBL2058653

SCHEMBL2058653

CN(CCCCl)Cc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.65
CARM1 Q86X55 1/20 0.60
PRMT6 Q96LA8 1/20 0.60
PRMT8 Q9NR22 1/20 0.60
LMNA P02545 1/20 0.57
TMEM97 Q5BJF2 2/20 0.54
MAOB P27338 4/20 0.53
MAOA P21397 1/20 0.53
TSHR P16473 2/20 0.51
ALDH1A1 P00352 1/20 0.50
ACHE P22303 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1593475 0.98 SIGMAR1 (0.62) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL11203747 0.94 SIGMAR1 (0.68) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL11872505 0.92 SIGMAR1 (0.71) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL2001215 0.88 CARM1 (0.64) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL1088446 0.87 SIGMAR1 (0.74) SIGMAR1CARM1PRMT6PRMT8LMNA
Hydrochloric Acid SCHEMBL394643 0.86 CARM1 (0.62) SIGMAR1CARM1PRMT6PRMT8LMNA
Hydrochloric Acid SCHEMBL11109064 0.86 CARM1 (0.62) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL29733117 0.85 SIGMAR1 (0.85) SIGMAR1CARM1PRMT6PRMT8LMNA
SCHEMBL7225346 0.85 SIGMAR1 (0.85) SIGMAR1CARM1PRMT6PRMT8LMNA
Hydrochloric Acid SCHEMBL1087168 0.85 SIGMAR1 (0.71) SIGMAR1CARM1PRMT6PRMT8LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 200 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023099462-A1 AMINE-CONTAINING VINYLDISILOXANES IN THE MANUFACTURE OF ELASTOMERIC POLYMERS TRINSEO EUROPE GMBH (CH) 2023-06-08 WO disclosed
EP-4186911-A1 AMINE-CONTAINING VINYLDISILOXANES IN THE MANUFACTURE OF ELASTOMERIC POLYMERS Trinseo Europe GmbH (CH) 2023-05-31 EP disclosed
EP-3154934-B1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES UNIV LILLE (FR) 2021-04-14 EP disclosed
US-20210040034-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES UNIV LILLE II DROIT & SANTE (FR) 2021-02-11 US disclosed
US-10844008-B2 Compounds, pharmaceutical composition and their use in treating neurodegenerative diseases UNIVERSITE DE LILLE 2 DROIT ET SANTE (FR) 2020-11-24 US disclosed
CN-106795100-B Compound, pharmaceutical composition and its purposes in treatment neurodegenerative disease 里尔大学 2019-11-19 CN disclosed
US-20190092721-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES UNIVERSITE DE LILLE 2 DROIT ET SANTE (FR) 2019-03-28 US disclosed
US-10179761-B2 Compounds, pharmaceutical composition and their use in treating neurodegenerative diseases UNIVERSITE DE LILLE 2 DROIT ET SANTE (FR) 2019-01-15 US disclosed
CN-106795100-A Compound, pharmaceutical composition and its purposes in nerve degenerative diseases are treated 法国里尔第二大学 2017-05-31 CN disclosed
US-20170107174-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES UNIVERSITE DE LILLE (FR) 2017-04-20 US disclosed
US-4751223-A Antiinflammatory and analgesic aminoalkyl tetracyclic benzodiazepines HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-14 US disclosed
EP-0268793-A1 Aminoalkyl tetracyclic benzodiazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-06-01 EP disclosed
US-4728652-A VASODILATORS E. R. SQUIBB & SONS, INC. (US) 1988-03-01 US disclosed
EP-0236902-A1 1,2,3,4-tetrahydro-6-substituted-4-aryl(or heterocyclo)-3-substituted-2-thioxo (or oxo)-5-pyrimidinecarboxylic acids and esters E.R. Squibb & Sons, Inc. (US) 1987-09-16 EP disclosed
US-4684655-A 1,2,3,4-tetrahydro-6-substituted-4-aryl-3-substituted-2-thioxo(or oxo)-5-pyrimidinecarboxylic acids and esters and use thereof to lower blood pressure E. R. SQUIBB & SONS, INC. (US) 1987-08-04 US disclosed
EP-0202654-A2 5-Carboxy-1,4-dihydropyrimidine derivatives E.R. Squibb & Sons, Inc. (US) 1986-11-26 EP disclosed
US-4405623-A HYPOTENSIVE AGENTS, VASODILATORS MASAYUKI ISHIKAWA (JP) 1983-09-20 US disclosed
EP-0040793-A1 Novel quinazoline-dione compounds, process for production thereof and pharmaceutical use thereof Ishikawa, Masayuki (JP) 1981-12-02 EP disclosed
US-4232027-A ANTIINFLAMMATORY AGENTS E. R. SQUIBB & SONS, INC. (US) 1980-11-04 US disclosed
US-4021557-A BRONCHOSPASMOLYTICS BOEHRINGER INGELHEIM GMBH (DT) 1977-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210040034-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES MAPT, PSEN2, SNCA SIGMAR1 1439/4885CARM1 4151/4885PRMT6 4271/4885
US-10844008-B2 Compounds, pharmaceutical composition and their use in treating neurodegenerative diseases MAPT, PSEN2, SNCA SIGMAR1 1439/4885CARM1 4151/4885PRMT6 4271/4885
US-20170107174-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES MAPT, PSEN2, SNCA SIGMAR1 1439/4885CARM1 4151/4885PRMT6 4271/4885
US-20190092721-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITION AND THEIR USE IN TREATING NEURODEGENERATIVE DISEASES MAPT, PSEN2, SNCA SIGMAR1 1439/4885CARM1 4151/4885PRMT6 4271/4885
US-10179761-B2 Compounds, pharmaceutical composition and their use in treating neurodegenerative diseases MAPT, PSEN2, SNCA SIGMAR1 1439/4885CARM1 4151/4885PRMT6 4271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.