SCHEMBL20588488

SCHEMBL20588488

Cc1nc2n(C)ccc(=O)n2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 3/20 0.34
HSD17B10 Q99714 1/20 0.34
BRD4 O60885 1/20 0.33
TAF1 P21675 1/20 0.33
BRPF1 P55201 1/20 0.33
CREBBP Q92793 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM6A O15550 1/20 0.32
KDM4A O75164 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM5C P41229 1/20 0.32
KDM2B Q8NHM5 1/20 0.32
DOHH Q9BU89 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22627370 0.72 EGLN2 (0.36) HAVCR2HSD17B10BRD4TAF1BRPF1
SCHEMBL20587988 0.67 KDM4E (0.33) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL22071869 0.62 ADORA3 (0.36) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL26476552 0.62 DPP4 (0.33) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL15730362 0.60 ALDH1A1 (0.65) HSD17B10KDM4EALDH1A1L3MBTL1
SCHEMBL22302554 0.60 BRD4 (0.34) HAVCR2HSD17B10BRD4TAF1BRPF1
SCHEMBL12012176 0.60 HAVCR2 (0.41) HAVCR2HSD17B10KDM4EALDH1A1L3MBTL1
SCHEMBL19577292 0.59 CRBN (0.37) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL5510924 0.59
SCHEMBL439647 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018229683-A1 5,6-FUSED-BICYCLIC COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2018-12-20 WO disclosed