SCHEMBL20599370

SCHEMBL20599370

Clc1ncccc1-c1ncco1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.43
BRD4 O60885 1/20 0.41
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGDS O60760 1/20 0.40
ADRA1A P35348 4/20 0.39
ADRA1D P25100 3/20 0.39
LTA4H P09960 1/20 0.39
NPC1 O15118 6/20 0.38
RAB9A P51151 6/20 0.38
MAPT P10636 4/20 0.38
PKM P14618 1/20 0.38
ADRA2A P08913 2/20 0.38
ADRA1B P35368 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NFKB1 P19838 1/20 0.36
CASP3 P42574 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1919495 0.79 HPGDS (0.52) PIN1BRD4HPGDSADRA1AADRA1D
SCHEMBL739276 0.78 NPC1 (0.53) PIN1BRD4SMN1; SMN2HPGDSADRA1A
SCHEMBL30457886 0.78 NPC1 (0.53) PIN1BRD4SMN1; SMN2HPGDSADRA1A
SCHEMBL314058 0.78 TDP1 (0.42) PIN1BRD4HPGDSADRA1AADRA1D
SCHEMBL31734567 0.77 BRD4 (0.41) PIN1BRD4LMNASMN1; SMN2HPGDS
SCHEMBL30792106 0.77 MAP4K4 (0.44) PIN1BRD4HPGDSADRA1AADRA1D
SCHEMBL26259967 0.75 BRD4 (0.53) PIN1BRD4LMNASMN1; SMN2HPGDS
SCHEMBL24097956 0.73 BRD4 (0.41) PIN1BRD4HPGDSADRA1AADRA1D
SCHEMBL31571148 0.73 ALOX15 (0.46) BRD4SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL1600286 0.73 ALOX15 (0.46) BRD4SMN1; SMN2NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019000238-A1 5-(PYRIDIN-3-YL)OXAZOLE ALLOSTERIC MODULATORS OF M4 MUSCARINIC ACETYLCHOLINE RECEPTOR MERCK SHARP & DOHME CORP. (US) 2019-01-03 WO disclosed