SCHEMBL20599884

SCHEMBL20599884

Oc1ccc(-c2ccccc2Br)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.56
EP300 Q09472 2/20 0.45
KAT2B Q92831 2/20 0.45
KAT8 Q9H7Z6 2/20 0.45
HDAC3 O15379 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
LDHA P00338 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
POLB P06746 1/20 0.42
GRM2 Q14416 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CTSB P07858 1/20 0.38
CYP1A2 P05177 1/20 0.38
APP P05067 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30106400 1.00 IDO1 (0.56) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL13265824 0.83 IDO1 (0.81) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL442916 0.83 IDO1 (0.81) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL225430 0.77 IDO1 (0.68) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL29372744 0.77 IDO1 (0.68) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL2936933 0.77 ALDH1A1 (0.50) IDO1ALDH1A1MAPK1POLBKDM4E
SCHEMBL11504207 0.76 CYP1A2 (0.62) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL30827114 0.76 CYP1A2 (0.62) IDO1EP300KAT2BKAT8HDAC3
SCHEMBL358976 0.75 ALDH1A1 (0.67) IDO1ALDH1A1MAPK1KDM4EMAPT
SCHEMBL31295703 0.75 ALDH1A1 (0.67) IDO1ALDH1A1MAPK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11746283-B2 Silole and germole fused ring photochromic compounds TRANSITIONS OPTICAL, LTD. (IE) 2023-09-05 US disclosed
CN-110799514-B Silole and germacyclopentadiene fused ring photochromic compounds 光学转变有限公司 2023-01-31 CN disclosed
EP-3645540-B1 SILOLE AND GERMOLE FUSED RING PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL LTD (IE) 2021-11-03 EP disclosed
US-20200172798-A1 Silole and Germole Fused Ring Photochromic Compounds TRANSITIONS OPTICAL, LTD. (IE) 2020-06-04 US disclosed
EP-3645540-A1 SILOLE AND GERMOLE FUSED RING PHOTOCHROMIC COMPOUNDS Transitions Optical, Ltd. (IE) 2020-05-06 EP disclosed
CN-110799514-A Silole and germacyclopentadiene fused ring photochromic compounds 光学转变有限公司 2020-02-14 CN disclosed
WO-2019001724-A1 SILOLE AND GERMOLE FUSED RING PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL, LTD. (IE) 2019-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200172798-A1 Silole and Germole Fused Ring Photochromic Compounds CCNB2, SKP2, CCNB1 IDO1 1521/4885EP300 2849/4885KAT2B 1019/4885
US-11746283-B2 Silole and germole fused ring photochromic compounds CCNB2, SKP2, CCNB1 IDO1 1521/4885EP300 2849/4885KAT2B 1019/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.