SCHEMBL20599951

SCHEMBL20599951

O=c1cc(COCc2ccccc2)[nH]c(=O)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
YTHDC1 Q96MU7 1/20 0.50
GPR84 Q9NQS5 6/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TYMP P19971 2/20 0.43
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 1/20 0.42
UNG P13051 1/20 0.41
RAB9A P51151 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NSD2 O96028 1/20 0.41
ABL1 P00519 1/20 0.41
PPARG P37231 1/20 0.41
RIN1 Q13671 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
DAO P14920 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878921 0.84 SMN1; SMN2 (0.67) TSHRGPR84SMN1; SMN2ALDH1A1KMT2A
SCHEMBL1287276 0.79 SMN1; SMN2 (0.69) YTHDC1GPR84SMN1; SMN2TYMPTP53
SCHEMBL20599921 0.77 SMN1; SMN2 (0.57) TSHRGPR84SMN1; SMN2TYMPHSD17B10
SCHEMBL21234494 0.76 UNG (0.55) GPR84TYMPUNG
Dimethylamine SCHEMBL27691701 0.75 SMN1; SMN2 (0.63) YTHDC1GPR84SMN1; SMN2TYMPTP53
SCHEMBL20625702 0.74 TDP1 (0.53) GPR84SMN1; SMN2ALDH1A1UNGRAB9A
SCHEMBL14426642 0.73 RAB9A (0.72) TSHRYTHDC1GPR84SMN1; SMN2TYMP
SCHEMBL20625637 0.72 GPR84 (0.53) TSHRGPR84SMN1; SMN2HSD17B10UNG
SCHEMBL4625744 0.72 SMN1; SMN2 (0.56) TSHRYTHDC1GPR84SMN1; SMN2TYMP
SCHEMBL9222745 0.71 SMN1; SMN2 (0.41) TSHRYTHDC1GPR84SMN1; SMN2TYMP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019002407-A1 PROCESS FOR THE PREPARATION OF TIPIRACIL HYDROCHLORIDE AMNEAL PHARMACEUTICALS COMPANY GMBH (CH) 2019-01-03 WO disclosed